SCHEMBL7337972

SCHEMBL7337972

CC(C)(C)OC(=O)c1ncn2c1c(C(=O)N1CCCC1)cc1ccccc12

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 3/20 0.38
GABRG2 P18507 3/20 0.38
GABRB3 P28472 3/20 0.38
GABRA5 P31644 3/20 0.38
GABRA3 P34903 2/20 0.38
GABRA6 Q16445 1/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 1/20 0.38
GABRA2 P47869 1/20 0.38
GABRA4 P48169 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7329520 0.85 HSD17B10 (0.43) HPGDHSD17B10
SCHEMBL7332980 0.78 GABRA1 (0.40) GABRA1GABRG2GABRB3GABRA5HPGD
SCHEMBL7291196 0.71 PTPN2 (0.41) GABRA1GABRG2GABRB3GABRA5HPGD
SCHEMBL9599814 0.69 GABRA1 (0.47) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7335649 0.67 GABRA1 (0.39) GABRA1GABRG2GABRB3GABRA5
SCHEMBL7335647 0.67 GABRA1 (0.39) GABRA1GABRG2GABRB3GABRA5
SCHEMBL9075553 0.67
SCHEMBL9606957 0.67 GABRA5 (0.46) GABRA1GABRG2GABRB3GABRA5HPGD
SCHEMBL9077632 0.67
SCHEMBL9078291 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5935970-A Use of imidazo 1,5-a!quinolones as neuroprotective agents PHARMACIA & UPJOHN COMPANY (US) 1999-08-10 US claimed
US-RE35840-E Imidazo 1,5-a!quinolines for treatment of anxiety and sleep disorders PHARMACIA & UPJOHN COMPANY (US) 1998-07-07 US claimed
US-5594140-A Imidazo[1,5-A]quinolines for treatment of anxiety and sleep disorders THE UPJOHN COMPANY (US) 1997-01-14 US claimed
WO-1997000074-A1 USE OF IMIDAZO[1,5-a]QUINOLONES AS NEUROPROTECTIVE AGENTS PHARMACIA & UPJOHN COMPANY (US) 1997-01-03 WO claimed
EP-0729469-A1 IMIDAZO [1,5-a]QUINOLINES FOR TREATMENT OF ANXIETY AND SLEEP DISORDERS PHARMACIA & UPJOHN COMPANY (US) 1996-09-04 EP claimed
WO-1995014020-A1 IMIDAZO[1,5-a]QUINOLINES FOR TREATMENT OF ANXIETY AND SLEEP DISORDERS THE UPJOHN COMPANY (US) 1995-05-26 WO claimed