SCHEMBL7338294

SCHEMBL7338294

CC(C(=O)OCc1ccccc1)C(N)N1CCC(C(N)(OC=O)c2ccccc2N)CC1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.34
CYP2C19 P33261 1/20 0.34
PREP P48147 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
CHRM4 P08173 1/20 0.33
DPP4 P27487 2/20 0.33
DPP7 Q9UHL4 2/20 0.33
KCNH2 Q12809 1/20 0.33
CCR1 P32246 1/20 0.32
CSNK1A1 P48729 1/20 0.32
ACE2 Q9BYF1 1/20 0.32
CYP1A2 P05177 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6584997 0.87 UBE2M (0.35) PREPNPC1RAB9ADPP4DPP7
SCHEMBL6584489 0.80 HRH1 (0.42) PREPCCR1CYP1A2
SCHEMBL8547440 0.77 HTT (0.33) SMN1; SMN2CYP2C19PREPNPC1RAB9A
SCHEMBL6586315 0.74 DPP4 (0.37) SMN1; SMN2NPC1RAB9ADPP4DPP7
SCHEMBL6584617 0.68 HTT (0.36) SMN1; SMN2CYP2C19NPC1RAB9ADPP4
Tert-Butyl Formate SCHEMBL28751186 0.66 ITGB3 (0.43) CYP2C19DPP4DPP7KCNH2
SCHEMBL29061106 0.63 SMN1; SMN2 (0.66) SMN1; SMN2CYP2C19NPC1RAB9AHTT
SCHEMBL12640200 0.63 ALDH1A1 (0.64) NPC1RAB9A
SCHEMBL24974571 0.62 HRH3 (0.49) SMN1; SMN2CYP2C19NPC1RAB9AKCNH2
SCHEMBL13302682 0.62 ALDH1A1 (0.55) CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6002009-A Di-substituted 1,4-piperidine esters and amides having 5-HT4 antagonistic activity BOEHRINGER INGELHEIM ITALIA, S.P.A. (IT) 1999-12-14 US disclosed
WO-1996028424-A1 DI-SUBSTITUTED 1,4-PIPERIDINE ESTERS AND AMIDES HAVING 5-HT4 ANTAGONISTIC ACTIVITY BOEHRINGER INGELHEIM ITALIA S.P.A. (IT) 1996-09-19 WO disclosed