SCHEMBL7345470

SCHEMBL7345470

COc1ccc2c(c1)c(CNO)c(C)n2C(=O)c1ccc(Cl)cc1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 5/20 0.79
PTGS2 P35354 10/20 0.78
AKR1C3 P42330 3/20 0.78
CNR2 P34972 1/20 0.78
ALOX5 P09917 2/20 0.77
AKR1C2 P52895 2/20 0.77
MAPT P10636 2/20 0.77
KMT2A Q03164 2/20 0.77
NPSR1 Q6W5P4 2/20 0.77
KDM4E B2RXH2 1/20 0.77
MEN1 O00255 1/20 0.77
PTGES O14684 1/20 0.77
ABCC3 O15438 1/20 0.77
ABCC4 O15439 1/20 0.77
ABCB11 O95342 1/20 0.77
MT-CO2 P00403 1/20 0.77
LMNA P02545 1/20 0.77
ALB P02768 1/20 0.77
CYP1A2 P05177 1/20 0.77
ABCB1 P08183 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17384908 0.91 PTGS2 (0.76) PTGS1PTGS2AKR1C3CNR2ALOX5
SCHEMBL13653013 0.90 ALOX5 (0.79) PTGS1PTGS2AKR1C3CNR2ALOX5
SCHEMBL860853 0.89 PTGS2 (0.80) PTGS1PTGS2AKR1C3CNR2ALOX5
SCHEMBL4538035 0.89 PTGS1 (0.83) PTGS1PTGS2AKR1C3CNR2ALOX5
Oxametacin SCHEMBL24552 0.88 PTGS1 (1.00) PTGS1PTGS2AKR1C3CNR2ALOX5
Oxametacin SCHEMBL29378857 0.88 PTGS1 (1.00) PTGS1PTGS2AKR1C3CNR2ALOX5
SCHEMBL14086813 0.88 PTGS2 (1.00) PTGS1PTGS2AKR1C3CNR2ALOX5
SCHEMBL30426824 0.88 PTGS2 (1.00) PTGS1PTGS2AKR1C3CNR2ALOX5
SCHEMBL21119569 0.88 ALOX5 (0.75) PTGS1PTGS2AKR1C3CNR2ALOX5
SCHEMBL9040318 0.88 PTGS2 (0.78) PTGS1PTGS2AKR1C3CNR2ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112846-A Nonsteroidal antiinflammatory agents WARNER-LAMBERT COMPANY (US) 1992-05-12 US disclosed
US-5075330-A N-hydroxyamide, N-hydroxythioamide, N-hydroxyurea, and N-hydroxythiourea derivatives of selected NSAIDS as antiinflammatory agents WARNER-LAMBERT CO. (US) 1991-12-24 US disclosed
US-4981865-A N-hydroxyamide, N-hydroxythioamide, hydroxyurea, and N-hydroxythiourea derivatives of selected nsaids as antiinflammatory agents WARNER-LAMBERT CO. (US) 1991-01-01 US disclosed