SCHEMBL7345537

SCHEMBL7345537

CC(C)=C1Oc2cccc(OCC#CCN3CCC(NC(=O)c4ccc(C(F)(F)F)cc4)CC3)c2C1=O

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A5 Q9Y345 11/20 0.44
SCN1A P35498 1/20 0.41
SCN5A Q14524 1/20 0.41
SCN9A Q15858 1/20 0.41
DRD4 P21917 6/20 0.41
HTR2A P28223 3/20 0.41
DRD2 P14416 3/20 0.40
DRD3 P35462 1/20 0.40
HTR1A P08908 1/20 0.38
HTR7 P34969 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7352709 0.93 HTR7 (0.45) DRD4HTR2ADRD2DRD3HTR1A
SCHEMBL7356138 0.91 DRD4 (0.38) DRD4HTR1AHTR7
SCHEMBL7346919 0.87 UTS2R (0.42) DRD4HTR2ADRD2HTR1AHTR7
SCHEMBL6457611 0.87 SLC6A5 (0.51) SLC6A5SCN1ASCN5ASCN9ADRD4
SCHEMBL7346972 0.85 SLC6A5 (0.60) SLC6A5DRD4HTR2ADRD2
SCHEMBL7346054 0.84 CNR2 (0.40) HTR1AHTR7
SCHEMBL6466592 0.80 HTR7 (0.55) SLC6A5HTR2ADRD2DRD3HTR1A
SCHEMBL6458101 0.79 HTR7 (0.54) SLC6A5HTR2ADRD2DRD3HTR1A
SCHEMBL6462598 0.79 HTR7 (0.54) SLC6A5HTR2ADRD2DRD3HTR1A
SCHEMBL6462987 0.78 HTR7 (0.47) HTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6307051-B1 UROKINASE-TYPE PLASMINOGEN ACTIVATOR ANTAGONISTS AND HAVE ANTITUMOR AND ANTIMETASTATIC ACTIVITY. ROCHE DIAGNOSTICS GMBH (DE) 2001-10-23 US disclosed
EP-1026165-A1 O-substituted Hydroxycoumaranone derivatives as antitumor and antimetastatic agents Roche Diagnostics GmbH (DE) 2000-08-09 EP disclosed