SCHEMBL7347349

SCHEMBL7347349

Oc1ccc(-c2ccccc2Cc2ccc(CN3CCCC3)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 8/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C19 P33261 1/20 0.50
HRH4 Q9H3N8 1/20 0.50
OPRM1 P35372 2/20 0.45
OPRK1 P41145 2/20 0.45
KEAP1 Q14145 1/20 0.45
PTAFR P25105 2/20 0.44
DRD4 P21917 1/20 0.44
CD274 Q9NZQ7 2/20 0.44
CHKA P35790 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7348199 0.81 ESR1 (0.65) HRH3
SCHEMBL1071093 0.78 KEAP1 (0.55) KEAP1
SCHEMBL27768912 0.78 KEAP1 (0.60) KEAP1CD274
SCHEMBL322305 0.78 HRH3 (0.74) HRH3CYP2D6CYP2C19HRH4DRD4
SCHEMBL7440889 0.78 HRH3 (0.58) HRH3CYP2D6CYP2C19HRH4
SCHEMBL1888525 0.77 HRH3 (0.78) HRH3CYP2D6CYP2C19HRH4
Methane SCHEMBL8063684 0.75 HRH3 (0.75) HRH3CYP2D6CYP2C19HRH4
SCHEMBL7101510 0.72 LMNA (0.53) HRH3DRD4
SCHEMBL7442242 0.72 LTA4H (0.69) HRH3DRD4
Phenol SCHEMBL27575460 0.72 KEAP1 (0.50) KEAP1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993300-A4 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2002-07-31 EP disclosed
EP-0993300-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 2000-04-19 EP disclosed
WO-1998048798-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 1998-11-05 WO disclosed