SCHEMBL7348231

SCHEMBL7348231

O=C(Cc1cccc2ccccc12)N[C@@H](Cc1ccccc1)C(=O)CSCc1ccco1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C19 P33261 1/20 0.45
POLB P06746 2/20 0.44
PIN1 Q13526 1/20 0.43
LCK P06239 2/20 0.43
HPGD P15428 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
GAA P10253 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
GLA P06280 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
HRH4 Q9H3N8 1/20 0.40
CASP1 P29466 2/20 0.40
PSMB5 P28074 1/20 0.40
PKM P14618 1/20 0.39
MCHR1 Q99705 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7307336 0.92 PSMB5 (0.47) ALDH1A1CYP1A2CYP2C19LCKCASP1
SCHEMBL7342412 0.85 ALDH1A1 (0.49) ALDH1A1POLBLCKHPGDL3MBTL1
SCHEMBL7348676 0.84 POLB (0.52) ALDH1A1CYP1A2CYP2C19POLBHPGD
SCHEMBL7346557 0.81 CTSG (0.48) ALDH1A1POLBHPGDMAPTKMT2A
SCHEMBL7346551 0.81 CTSG (0.48) ALDH1A1POLBHPGDMAPTKMT2A
SCHEMBL7350634 0.81 ALDH1A1 (0.58) ALDH1A1CYP1A2CYP2C19POLBHPGD
SCHEMBL7342540 0.80 PSMB5 (0.47) ALDH1A1POLBHPGDGAAMAPT
SCHEMBL7343844 0.80 HPGD (0.53) ALDH1A1CYP2C19POLBHPGDL3MBTL1
SCHEMBL7342545 0.80 PSMB5 (0.47) ALDH1A1POLBHPGDGAAMAPT
SCHEMBL7348935 0.80 ALDH1A1 (0.41) ALDH1A1CYP1A2CYP2C19POLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0603873-B1 Aminoketone derivatives MITSUBISHI CHEM CORP (JP) 1998-04-15 EP disclosed
US-5424325-A Inibitors of thiol protease and may be used as therapeutic agents for treating muscular dystrophy, cataracts, strokes MITSUBISHI KASEI CORPORATION (JP) 1995-06-13 US disclosed
EP-0603873-A1 Aminoketone derivatives Mitsubishi Chemical Corporation (JP) 1994-06-29 EP disclosed