SCHEMBL7348446

SCHEMBL7348446

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCN2Cc3ccccc3C2)C1c1cnc2ccccc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.46
PDE1C Q14123 4/20 0.46
CACNA1F O60840 2/20 0.43
CACNA1D Q01668 2/20 0.43
CACNA1S Q13698 2/20 0.43
CACNA1C Q13936 2/20 0.43
ADRA1A P35348 5/20 0.43
ADRA2A P08913 4/20 0.43
ADRA2B P18089 4/20 0.43
ADRA2C P18825 4/20 0.43
ADRA1D P25100 4/20 0.43
ADRA1B P35368 4/20 0.43
ABCB1 P08183 2/20 0.43
MAPT P10636 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
MEN1 O00255 1/20 0.43
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
CHRM2 P08172 1/20 0.43
CYP3A4 P08684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7346339 0.84 HSD17B10 (0.59) ADORA3PDE1CCACNA1FCACNA1DCACNA1S
SCHEMBL7348450 0.83 ADORA3 (0.56) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7347758 0.82 GAA (0.52) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7348456 0.81 ADORA3 (0.43) ADORA3PDE1CCACNA1FCACNA1DCACNA1S
SCHEMBL7345495 0.80 POLB (0.58) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7349297 0.80 CACNA1B (0.57) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7343709 0.80 CACNA1B (0.52) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7341777 0.80 CACNA1F (0.63) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7344603 0.80 KDM4E (0.67) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7344610 0.79 HSD17B10 (0.52) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed