SCHEMBL7350412

SCHEMBL7350412

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCC2NCc3ccccc32)C1c1c[nH]c2ccccc12

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE1C Q14123 1/20 0.65
GAA P10253 2/20 0.42
ADORA3 P0DMS8 5/20 0.42
CYP2C9 P11712 4/20 0.42
CYP1A2 P05177 4/20 0.42
ABCB11 O95342 4/20 0.42
KDM4E B2RXH2 3/20 0.42
CYP3A4 P08684 3/20 0.42
CYP2C19 P33261 3/20 0.42
KMT2A Q03164 3/20 0.42
HIF1A Q16665 3/20 0.42
HSD17B10 Q99714 3/20 0.42
LMNA P02545 3/20 0.42
SCN1A P35498 3/20 0.42
SCN5A Q14524 3/20 0.42
SCN2A Q99250 3/20 0.42
SCN3A Q9NY46 3/20 0.42
NR1I2 O75469 3/20 0.42
MEN1 O00255 2/20 0.42
NR3C1 P04150 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7349531 0.84 ADORA3 (0.55) GAAADORA3CYP2C9CYP1A2ABCB11
SCHEMBL7343553 0.84 ADORA3 (0.45) GAAADORA3CYP2C9CYP1A2ABCB11
SCHEMBL7348034 0.84 CACNA1C (0.46) GAAADORA3CYP2C9CYP1A2ABCB11
SCHEMBL7342398 0.83 ADORA3 (0.43) PDE1CGAAADORA3CYP2C9CYP1A2
SCHEMBL7351371 0.81 CYP1A2 (0.66) ADORA3CYP2C9CYP1A2ABCB11KDM4E
SCHEMBL7350408 0.81 PDE1C (0.69) PDE1CGAAADORA3CYP2C9CYP1A2
SCHEMBL10744175 0.80 ALDH1A1 (0.51) GAAADORA3KDM4EKMT2AHSD17B10
SCHEMBL7349721 0.80 KDM4E (0.62) GAAADORA3CYP2C9CYP1A2KDM4E
SCHEMBL7344608 0.80 KDM4E (0.62) GAAADORA3CYP2C9CYP1A2ABCB11
SCHEMBL7344616 0.80 CACNA1B (0.49) ADORA3KDM4EHSD17B10LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed