SCHEMBL7350906

SCHEMBL7350906

COc1cccc(N2CCN(CCCCN3C(=O)NCC3c3cccc(Cl)c3)CC2)c1

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.67
HTR1A P08908 4/20 0.52
ABCB1 P08183 2/20 0.51
MAPT P10636 1/20 0.51
TSHR P16473 1/20 0.51
ALDH1A1 P00352 1/20 0.50
DRD4 P21917 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7343619 0.91 KCNH2 (0.54) KCNH2
SCHEMBL7347718 0.91 KCNH2 (0.53) KCNH2HTR1AMAPTDRD4
SCHEMBL7353705 0.87 KCNH2 (0.52) KCNH2HTR1A
SCHEMBL7343246 0.84 ADRA1A (0.55) HTR1AALDH1A1
SCHEMBL4524281 0.82 KCNH2 (1.00) KCNH2HTR1AABCB1MAPTTSHR
SCHEMBL7355250 0.79 HTR1A (0.52) HTR1AMAPT
SCHEMBL13711973 0.78 KCNH2 (0.87) KCNH2ABCB1MAPTTSHRALDH1A1
SCHEMBL7347383 0.76 SLC6A3 (0.43)
SCHEMBL7344857 0.75 KCNH2 (0.52) KCNH2HTR1ADRD4
SCHEMBL7350903 0.75 KCNH2 (0.76) KCNH2HTR1AMAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536279-A1 SUBSTITUTED 1-(ALKOXYPHENYL)PIPERAZINES WITH CNS AND ANTIHYPERTENSIVE ACTIVITY THE UPJOHN COMPANY (US) 1993-04-14 EP disclosed
WO-1992000282-A1 SUBSTITUTED 1-(ALKOXYPHENYL)PIPERAZINES WITH CNS AND ANTIHYPERTENSIVE ACTIVITY THE UPJOHN COMPANY (US) 1992-01-09 WO disclosed