SCHEMBL7351045

SCHEMBL7351045

CC(C)=C1Oc2cccc(OCCNCCN3CCC(NC(=O)c4ccc(Cl)c(Cl)c4)CC3)c2C1=O

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 5/20 0.47
HTR1A P08908 2/20 0.45
UTS2R Q9UKP6 11/20 0.44
SSTR5 P35346 1/20 0.40
KCNH2 Q12809 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6381981 0.93 HTR7 (0.49) HTR7HTR1AUTS2RSSTR5KCNH2
SCHEMBL7348639 0.92 HTR7 (0.44) HTR7HTR1AUTS2RSSTR5KCNH2
SCHEMBL7347807 0.89 HTR7 (0.53) HTR7HTR1ASSTR5
SCHEMBL7351795 0.89 HTR7 (0.44) HTR7HTR1AUTS2R
SCHEMBL6823392 0.87 HTR7 (0.49) HTR7HTR1AUTS2RACHE
SCHEMBL6824342 0.86 HTR7 (0.43) HTR7HTR1AUTS2RSSTR5KCNH2
SCHEMBL6820561 0.86 UTS2R (0.45) HTR7HTR1AUTS2RSSTR5KCNH2
SCHEMBL6462162 0.86 MCHR1 (0.43) HTR7HTR1AUTS2RSSTR5KCNH2
SCHEMBL6462165 0.86 MCHR1 (0.43) HTR7HTR1AUTS2RSSTR5KCNH2
SCHEMBL6824741 0.85 HTR7 (0.47) HTR7HTR1AUTS2RSSTR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6307051-B1 UROKINASE-TYPE PLASMINOGEN ACTIVATOR ANTAGONISTS AND HAVE ANTITUMOR AND ANTIMETASTATIC ACTIVITY. ROCHE DIAGNOSTICS GMBH (DE) 2001-10-23 US disclosed
EP-1026165-A1 O-substituted Hydroxycoumaranone derivatives as antitumor and antimetastatic agents Roche Diagnostics GmbH (DE) 2000-08-09 EP disclosed