SCHEMBL7355372

SCHEMBL7355372

COC(=O)C(Cc1cccc2ccccc12)(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.50
CTSK P43235 2/20 0.50
ATM Q13315 1/20 0.43
NQO2 P16083 1/20 0.42
SSTR4 P31391 1/20 0.42
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 1/20 0.41
PTPRB P23467 1/20 0.41
GAA P10253 2/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TDP1 Q9NUW8 2/20 0.40
TACR1 P25103 1/20 0.40
CASR P41180 1/20 0.39
ACHE P22303 1/20 0.39
CTSL P07711 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7352587 0.93 CTSS (0.54) CTSSCTSKATMNQO2SSTR4
SCHEMBL9556336 0.90 CTSS (0.44) CTSSCTSKATMNQO2SSTR4
SCHEMBL9848710 0.77 ATM (0.48) CTSSCTSKATMSSTR4KDM4E
SCHEMBL8392933 0.75 ALDH1A1 (0.51) CTSSCTSKATMALDH1A1PTPRB
SCHEMBL16009313 0.74 CTSK (0.37) CTSSCTSKNQO2PTPRBCTSL
SCHEMBL27487742 0.74 CTSS (0.47) CTSSCTSKATMNQO2SSTR4
SCHEMBL9848642 0.74 ATM (0.52) ATMSSTR4KDM4EALDH1A1MEN1
SCHEMBL4600435 0.73 CTSS (0.76) CTSSCTSKCTSL
SCHEMBL613640 0.73 CTSS (0.76) CTSSCTSKCTSL
SCHEMBL29401990 0.73 CTSS (0.76) CTSSCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258362-A Enzyme inhibitors, amides with oxetane ring ABBOTT LABORATORIES (US) 1993-11-02 US disclosed
WO-1992022313-A1 RENIN INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-12-23 WO disclosed