SCHEMBL7356525

SCHEMBL7356525

COc1cc(OC2CCN(OC(C)(C)C)C(=C=O)C2)ccc1C(=[N+]=[N-])C(=O)C(=[N+]=[N-])c1ccc(OC2CCN(OC(C)(C)C)C(=C=O)C2)cc1OC

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.34
OXTR P30559 4/20 0.33
ALDH1A1 P00352 1/20 0.33
AVPR2 P30518 1/20 0.33
AVPR1A P37288 1/20 0.33
KDM2B Q8NHM5 3/20 0.32
RAB9A P51151 1/20 0.32
GPR6 P46095 1/20 0.32
PARP15 Q460N3 1/20 0.32
PARP10 Q53GL7 1/20 0.32
ACACB O00763 1/20 0.31
GPR119 Q8TDV5 3/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
HRH3 Q9Y5N1 2/20 0.31
HSD11B1 P28845 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7397848 0.84 GPR6 (0.33) ALDH1A1GPR6GPR119HSD11B1
SCHEMBL3563776 0.80 GRIK1 (0.43) ALDH1A1KDM2BRAB9AGPR6PDE4A
SCHEMBL7356519 0.80 GPR119 (0.49) ALDH1A1GPR119PDE4APDE4BPDE4C
SCHEMBL3554378 0.79 MEN1 (0.37) ALDH1A1KDM2BRAB9AGPR6PDE4B
SCHEMBL8094956 0.78 LIPG (0.38) GPR119HRH3
SCHEMBL9013863 0.73 GPR119 (0.38) GPR119HRH3
SCHEMBL7333820 0.73 OXTR (0.41) OXTRALDH1A1AVPR2AVPR1AACACB
SCHEMBL7333661 0.72 OXTR (0.42) OXTRALDH1A1AVPR2AVPR1AACACB
SCHEMBL8088578 0.72 EPHX2 (0.40) GPR119HRH3
SCHEMBL7335906 0.72 OXTR (0.37) OXTRGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0805681-A4 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1998-05-06 EP disclosed
EP-0805681-A1 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1997-11-12 EP disclosed
WO-1996022775-A1 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1996-08-01 WO disclosed