SCHEMBL7356908

SCHEMBL7356908

N[C@H](CC1CCCCC1)C(O)C(=O)NCc1cccc2ccccc12

nearest known ligand 0.70

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 15/20 0.70
METAP1 P53582 9/20 0.70
CHRNB2 P17787 1/20 0.50
CHRNB4 P30926 1/20 0.50
CHRNA3 P32297 1/20 0.50
CHRNA4 P43681 1/20 0.50
GRIN1 Q05586 1/20 0.50
GRIN2A Q12879 1/20 0.50
GRM1 Q13255 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7355712 0.99 METAP2 (0.69) METAP2METAP1CHRNB2CHRNB4CHRNA3
SCHEMBL23710399 0.86 METAP2 (0.53) METAP2METAP1CHRNB2CHRNB4CHRNA3
SCHEMBL14984962 0.85 METAP2 (0.55) METAP2METAP1CHRNB2CHRNB4CHRNA3
SCHEMBL7354275 0.84 METAP2 (0.63) METAP2METAP1
SCHEMBL7362423 0.84 METAP2 (0.63) METAP2METAP1
SCHEMBL19309026 0.83 METAP2 (0.53) METAP2METAP1CHRNB2CHRNB4CHRNA3
SCHEMBL12022117 0.83 METAP2 (0.53) METAP2METAP1CHRNB2CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL7352923 0.83 METAP2 (0.62) METAP2METAP1
SCHEMBL5534127 0.83 CHRNB2 (0.50) METAP2METAP1CHRNB2CHRNB4CHRNA3
SCHEMBL7358087 0.81 METAP2 (0.60) METAP2METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
WO-2017123603-A1 TREATMENT FOR TUMORS DRIVEN BY METABOLIC DYSFUNCTION SYNDEVRX, INC. (US) 2017-07-20 WO disclosed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP disclosed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed