SCHEMBL7357973

SCHEMBL7357973

Cc1[nH]c2ccc(N)cc2c1C(=O)CCc1ccc(C#N)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
USP14 P54578 2/20 0.39
FFAR1 O14842 4/20 0.38
ESR1 P03372 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
MAP2 P11137 1/20 0.37
KMT2A Q03164 3/20 0.36
MITF O75030 1/20 0.36
LMNA P02545 1/20 0.36
RAB9A P51151 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SLC5A1 P13866 1/20 0.36
SLC5A2 P31639 1/20 0.36
GAA P10253 1/20 0.36
TBXAS1 P24557 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7424087 0.83 ALDH1A1 (0.47) ALDH1A1FFAR1ESR1CYP1A2CYP3A4
SCHEMBL7362233 0.82 ALDH1A1 (0.47) ALDH1A1ESR1CYP1A2CYP3A4CYP2C9
SCHEMBL7353853 0.81 ALDH1A1 (0.48) ALDH1A1ESR1CYP1A2CYP3A4CYP2C9
SCHEMBL7358998 0.78 USP14 (0.40) ALDH1A1USP14LMNAGAAMAPT
SCHEMBL7354262 0.78 PTGS1 (0.42) ALDH1A1USP14FFAR1ESR1CYP1A2
SCHEMBL7350830 0.77 TUBB1 (0.42) ALDH1A1USP14FFAR1ESR1CYP1A2
SCHEMBL7361052 0.76 CXCR2 (0.36) FFAR1CYP2C9MAP2CXCR2
SCHEMBL7361844 0.75 ALDH1A1 (0.46) ALDH1A1FFAR1ESR1CYP1A2CYP3A4
SCHEMBL7362067 0.72 F2 (0.49) ALDH1A1KMT2AMITFLMNARAB9A
SCHEMBL7358200 0.71 USP14 (0.41) ALDH1A1USP14FFAR1KMT2AMITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999028297-A1 SUBSTITUTED INDOLES, HAVING A THROMBIN INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-10 WO disclosed