SCHEMBL7350830

SCHEMBL7350830

Cc1[nH]c2cc(OC(=O)O)ccc2c1C(=O)CCc1ccc(C#N)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 1/20 0.42
ESR1 P03372 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPT P10636 2/20 0.40
MITF O75030 1/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
POLB P06746 1/20 0.38
FFAR1 O14842 2/20 0.38
ALDH1A1 P00352 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
SLC5A1 P13866 3/20 0.38
SLC5A2 P31639 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7424087 0.92 ALDH1A1 (0.47) ESR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7362233 0.83 ALDH1A1 (0.47) ESR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7353853 0.82 ALDH1A1 (0.48) ESR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7354262 0.80 PTGS1 (0.42) ESR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7361844 0.78 ALDH1A1 (0.46) ESR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7357973 0.77 ALDH1A1 (0.41) ESR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7358998 0.72 USP14 (0.40) ALOX15MAPTPOLBALDH1A1GAA
SCHEMBL7358416 0.71 PLA2G4A (0.38) FFAR1ALDH1A1FFAR4RAB9AKDM4E
SCHEMBL7357018 0.69 ALOX15 (0.43) ESR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7357066 0.68 KDM4E (0.42) MAPTALDH1A1RAB9AKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999028297-A1 SUBSTITUTED INDOLES, HAVING A THROMBIN INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-10 WO disclosed