SCHEMBL7358018

SCHEMBL7358018

N#C/N=C(\Nc1ccc(N)nc1)NC1(c2ccccc2)CCC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 2/20 0.35
HDAC3 O15379 4/20 0.34
HDAC1 Q13547 3/20 0.34
HDAC2 Q92769 3/20 0.34
HDAC6 Q9UBN7 3/20 0.34
NCOR2 Q9Y618 1/20 0.34
DPP4 P27487 1/20 0.32
TACR3 P29371 2/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
NAMPT P43490 2/20 0.31
OPRM1 P35372 1/20 0.30
OPRL1 P41146 1/20 0.30
BRAF P15056 1/20 0.30
CCKBR P32239 1/20 0.30
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7358020 1.00 VNN1 (0.35) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL8439682 0.89 VNN1 (0.36) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL7363327 0.83 VNN1 (0.35) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL7363331 0.83 VNN1 (0.35) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL7357917 0.82 P2RX7 (0.41) NAMPTMEN1NPC1ALDH1A1RAB9A
SCHEMBL13949283 0.82 P2RX7 (0.41) NAMPTMEN1NPC1ALDH1A1RAB9A
SCHEMBL4259491 0.82 P2RX7 (0.41) NAMPTMEN1NPC1ALDH1A1RAB9A
SCHEMBL8619031 0.82 HDAC3 (0.33) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL7354766 0.82 HDAC3 (0.33) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL7362655 0.82 VNN1 (0.34) VNN1HDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655057-B1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS UPJOHN CO (US) 1997-09-17 EP claimed
US-5567722-A DIURETICS THE UPJOHN COMPANY (US) 1996-10-22 US claimed
EP-0655057-A1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS. UPJOHN CO (US) 1995-05-31 EP claimed
WO-1994004500-A1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS THE UPJOHN COMPANY (US) 1994-03-03 WO claimed
EP-0655057-B1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS UPJOHN CO (US) 1997-09-17 EP disclosed
US-5567722-A DIURETICS THE UPJOHN COMPANY (US) 1996-10-22 US disclosed
EP-0655057-A1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS. UPJOHN CO (US) 1995-05-31 EP disclosed
WO-1994004500-A1 CYANOGUANIDINES AS POTASSIUM CHANNEL BLOCKERS THE UPJOHN COMPANY (US) 1994-03-03 WO disclosed