SCHEMBL8439682

SCHEMBL8439682

N#CN=C(Nc1cnc(N)nc1)NC1(c2ccccc2)CCC1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 2/20 0.36
HDAC3 O15379 4/20 0.35
HDAC1 Q13547 3/20 0.35
HDAC2 Q92769 3/20 0.35
HDAC6 Q9UBN7 3/20 0.35
DPP4 P27487 1/20 0.33
TACR3 P29371 2/20 0.32
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
ALOX5AP P20292 1/20 0.32
OPRM1 P35372 1/20 0.31
OPRL1 P41146 1/20 0.31
SSTR4 P31391 1/20 0.31
MAPK1 P28482 1/20 0.31
SCN9A Q15858 1/20 0.31
NCOR2 Q9Y618 1/20 0.31
MAPKAPK2 P49137 1/20 0.31
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7358018 0.89 VNN1 (0.35) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL7358020 0.89 VNN1 (0.35) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL7363331 0.85 VNN1 (0.35) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL7363327 0.85 VNN1 (0.35) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL7362657 0.84 VNN1 (0.34) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL7362655 0.84 VNN1 (0.34) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL7357917 0.82 P2RX7 (0.41) MAPK1
SCHEMBL13949283 0.82 P2RX7 (0.41) MAPK1
SCHEMBL4259491 0.82 P2RX7 (0.41) MAPK1
SCHEMBL8619031 0.79 HDAC3 (0.33) VNN1HDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0703904-B1 PYRIMIDINE CYANOGUANIDINES AS K-CHANNEL BLOCKERS UPJOHN CO (US) 1999-02-24 EP claimed
US-5633374-A Pyrimidine, cyanoguanidines as K-channel blockers THE UPJOHN COMPANY (US) 1997-05-27 US claimed
EP-0703904-B1 PYRIMIDINE CYANOGUANIDINES AS K-CHANNEL BLOCKERS UPJOHN CO (US) 1999-02-24 EP disclosed
US-5633374-A Pyrimidine, cyanoguanidines as K-channel blockers THE UPJOHN COMPANY (US) 1997-05-27 US disclosed