SCHEMBL7359486

SCHEMBL7359486

COc1ccc(CCC2(NCCC(=O)Nc3ccc(OC)c(OC)c3)CC2)cc1OC

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
NPSR1 Q6W5P4 2/20 0.50
LMNA P02545 4/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
HDAC1 Q13547 2/20 0.48
HDAC2 Q92769 2/20 0.48
CNR1 P21554 1/20 0.48
GAA P10253 1/20 0.47
PKM P14618 1/20 0.47
HTT P42858 1/20 0.47
EPHX2 P34913 1/20 0.47
POLB P06746 2/20 0.47
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
THRB P10828 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18760165 0.81 NPC1 (0.67) NPC1RAB9ANPSR1LMNASMN1; SMN2
SCHEMBL9775789 0.76 ALDH1A1 (0.58) NPC1RAB9ANPSR1LMNASMN1; SMN2
SCHEMBL23121264 0.72 NPC1 (0.62) NPC1RAB9ANPSR1LMNASMN1; SMN2
SCHEMBL7359470 0.72 NPSR1 (0.56) NPC1RAB9ANPSR1LMNASMN1; SMN2
SCHEMBL7335367 0.72 NPC1 (0.55) NPC1RAB9ANPSR1LMNASMN1; SMN2
SCHEMBL21852785 0.71 NPC1 (0.64) NPC1RAB9ANPSR1SMN1; SMN2HTT
SCHEMBL7355352 0.71 LMNA (0.56) NPC1RAB9ANPSR1LMNASMN1; SMN2
SCHEMBL7359187 0.71 KMT2A (0.58) NPC1RAB9ALMNASMN1; SMN2HDAC1
SCHEMBL7360125 0.71 NPC1 (0.55) NPC1RAB9ALMNASMN1; SMN2HDAC1
SCHEMBL7959722 0.70 NPC1 (0.63) NPC1RAB9ANPSR1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0852142-A1 Diamines in the treatment of arrhythmia SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1998-07-08 EP disclosed
EP-0639973-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1995-03-01 EP disclosed
WO-1993023024-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1993-11-25 WO disclosed