SCHEMBL7360094

SCHEMBL7360094

CCN(Cc1ccc(Cl)cc1Cl)C(=O)C(O)[C@H](N)CC1CCCCC1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 10/20 0.60
METAP1 P53582 5/20 0.60
SLC6A2 P23975 5/20 0.41
SLC6A4 P31645 5/20 0.41
CYP2D6 P10635 1/20 0.41
KCNH2 Q12809 1/20 0.41
PYGL P06737 1/20 0.39
AGTR2 P50052 1/20 0.39
SLC6A3 Q01959 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7353362 0.77 METAP2 (0.80) METAP2METAP1
Hydrochloric Acid SCHEMBL7509007 0.76 METAP2 (0.79) METAP2METAP1
SCHEMBL7361793 0.75 METAP2 (1.00) METAP2METAP1
Hydrochloric Acid SCHEMBL7353187 0.74 METAP2 (0.98) METAP2METAP1
SCHEMBL6561605 0.74 METAP2 (0.64) METAP2METAP1SLC6A2SLC6A4KCNH2
SCHEMBL7358163 0.72 METAP2 (0.67) METAP2METAP1
SCHEMBL6934858 0.69 METAP2 (0.46) METAP2METAP1PYGL
SCHEMBL6485894 0.69 METAP2 (0.84) METAP2METAP1
SCHEMBL6564599 0.69 METAP2 (0.64) METAP2METAP1SLC6A2SLC6A4SLC6A3
SCHEMBL7357040 0.69 METAP2 (0.52) METAP2METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US disclosed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP disclosed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed