SCHEMBL7360923

SCHEMBL7360923

N#Cc1ccc(CCCn2ccc3cc([N+](=O)[O-])ccc32)cc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 3/20 0.52
KCNH2 Q12809 2/20 0.52
RORC P51449 1/20 0.45
AR P10275 1/20 0.41
P2RX7 Q99572 1/20 0.40
SIGMAR1 Q99720 1/20 0.39
PLG P00747 1/20 0.39
PLAU P00749 1/20 0.39
CYP19A1 P11511 1/20 0.39
PKM P14618 1/20 0.38
HTR7 P34969 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7362873 0.80 RORC (0.44) KCNJ1KCNH2RORCP2RX7PLG
SCHEMBL2846720 0.77 PKM (0.62) RORCSIGMAR1CYP19A1PKM
SCHEMBL23902730 0.76 GLS (0.46) PLGPLAUCYP19A1HTR7
SCHEMBL2479169 0.76 HTR7 (0.47) PLGPLAUCYP19A1HTR7
SCHEMBL2263041 0.76 GLS (0.46) PLGPLAUCYP19A1PKMHTR7
SCHEMBL30241520 0.76 GLS (0.46) PLGPLAUCYP19A1HTR7
SCHEMBL6637649 0.76 KCNJ1 (0.53) KCNJ1KCNH2CYP19A1PKM
SCHEMBL9640859 0.76 KCNH2 (0.68) KCNJ1KCNH2SIGMAR1CYP19A1
SCHEMBL7357276 0.76 KRAS (0.52) RORCARPKM
SCHEMBL10430002 0.75 PLG (0.46) PLGPLAUCYP19A1HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999028297-A1 SUBSTITUTED INDOLES, HAVING A THROMBIN INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-10 WO disclosed