SCHEMBL7361014

SCHEMBL7361014

CC1CC(=O)c2c(S(C)(=O)=O)ccc(-c3cccc[n+]3[O-])c2C1

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 9/20 0.64
GABRB3 P28472 9/20 0.64
GABRA5 P31644 9/20 0.64
GABRA3 P34903 9/20 0.64
GABRA2 P47869 9/20 0.64
GABRA1 P14867 8/20 0.37
BRD4 O60885 3/20 0.34
STAT3 P40763 1/20 0.34
CSNK2A2 P19784 3/20 0.33
CSNK2B P67870 3/20 0.33
CSNK2A1 P68400 3/20 0.33
ABCG2 Q9UNQ0 3/20 0.33
CSNK2A3 Q8NEV1 1/20 0.33
EDNRB P24530 1/20 0.31
EDNRA P25101 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7349704 0.78 GABRG2 (0.74) GABRG2GABRB3GABRA5GABRA3GABRA2
SCHEMBL7358332 0.74 GABRG2 (0.67) GABRG2GABRB3GABRA5GABRA3GABRA2
SCHEMBL7354097 0.74 GABRG2 (0.67) GABRG2GABRB3GABRA5GABRA3GABRA2
SCHEMBL15093571 0.57 PNMT (0.40) BRD4STAT3
SCHEMBL16632833 0.57 PKM (0.42)
SCHEMBL29727517 0.56 LMNA (0.52) GABRG2GABRB3GABRA5GABRA3GABRA2
SCHEMBL871319 0.56 LMNA (0.52) GABRG2GABRB3GABRA5GABRA3GABRA2
SCHEMBL19865239 0.56 ACHE (0.41)
SCHEMBL4906168 0.55 IDO1 (0.41) GABRG2GABRB3GABRA5GABRA3GABRA2
SCHEMBL7360811 0.55 GABRG2 (0.71) GABRG2GABRB3GABRA5GABRA3GABRA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156761-A Substituted tetralone derivatives for enhancing cognition MERCK SHARPE & DOHME LIMITED (GB) 2000-12-05 US disclosed