SCHEMBL7362435

SCHEMBL7362435

CC(C)(NC(=O)c1ccc(C#N)cc1Cl)C(C(=O)N1CCC(CC(=O)OCc2ccccc2)CC1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.41
ITGA2B P08514 2/20 0.41
YAP1 P46937 9/20 0.40
MGLL Q99685 1/20 0.37
CHRM4 P08173 3/20 0.36
CCR1 P32246 1/20 0.36
CCL5 P13501 1/20 0.35
CCR5 P51681 1/20 0.35
P2RX7 Q99572 1/20 0.35
MCHR1 Q99705 1/20 0.35
CCKBR P32239 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7836339 0.88 YAP1 (0.44) ITGB3ITGA2BYAP1CHRM4P2RX7
SCHEMBL7835873 0.83 YAP1 (0.41) YAP1CHRM4P2RX7CCKBR
SCHEMBL7833217 0.83 GRIN2B (0.42) YAP1CHRM4P2RX7
SCHEMBL7357897 0.83 YAP1 (0.46) YAP1CHRM4P2RX7
SCHEMBL7839324 0.82 ITGB3 (0.44) ITGB3ITGA2BYAP1MGLLCHRM4
SCHEMBL7836103 0.80 CTSG (0.43) ITGB3ITGA2BYAP1CHRM4
SCHEMBL7833800 0.79 YAP1 (0.44) ITGB3ITGA2BYAP1CHRM4P2RX7
SCHEMBL7833534 0.78 YAP1 (0.43) ITGB3ITGA2BYAP1CHRM4CCR1
SCHEMBL7837038 0.78 ITGB3 (0.53) ITGB3ITGA2B
SCHEMBL7835452 0.78 PRSS1 (0.44) ITGB3ITGA2BYAP1CHRM4CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800516-B1 FIBRINOGEN RECEPTOR ANTAGONISTS HAVING SUBSTITUTED (b)-AMINO ACID RESIDUES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME NIPPON STEEL CORP (JP) 2001-09-19 EP disclosed
US-5866592-A Fibrinogen receptor antagonist and pharmaceutical compositions comprising the same NIPPON STEEL CORPORATION (JP) 1999-02-02 US disclosed
WO-1996020172-A1 FIBRINOGEN RECEPTOR ANTAGONISTS HAVING SUBSTITUTED β-AMINO ACID RESIDUES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME NIPPON STEEL CORPORATION (JP) 1996-07-04 WO disclosed