SCHEMBL7833217

SCHEMBL7833217

CC(C)(NC(=O)c1ccc(C#N)cc1)C(C(=O)N1CCC(CC(=O)OCc2ccccc2)CC1)c1ccncc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 5/20 0.42
CYP2D6 P10635 4/20 0.42
CYP2C9 P11712 4/20 0.42
YAP1 P46937 3/20 0.41
CHRM4 P08173 3/20 0.41
CCR3 P51677 1/20 0.39
PRSS1 P07477 2/20 0.39
CTSG P08311 2/20 0.39
CTRB1 P17538 2/20 0.39
CMA1 P23946 2/20 0.39
CYP3A4 P08684 3/20 0.38
P2RX7 Q99572 1/20 0.37
PRKAB2 O43741 1/20 0.37
PRKAG1 P54619 1/20 0.37
PRKAA2 P54646 1/20 0.37
PRKAA1 Q13131 1/20 0.37
PRKAG3 Q9UGI9 1/20 0.37
PRKAG2 Q9UGJ0 1/20 0.37
PRKAB1 Q9Y478 1/20 0.37
F2 P00734 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7836339 0.94 YAP1 (0.44) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7835873 0.91 YAP1 (0.41) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7357897 0.90 YAP1 (0.46) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7839324 0.88 ITGB3 (0.44) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7833800 0.86 YAP1 (0.44) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7836103 0.86 CTSG (0.43) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7833534 0.86 YAP1 (0.43) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7835452 0.84 PRSS1 (0.44) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7362435 0.83 ITGB3 (0.41) YAP1CHRM4P2RX7
SCHEMBL7835970 0.83 YAP1 (0.41) YAP1CHRM4CCR3PRSS1CTSG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800516-B1 FIBRINOGEN RECEPTOR ANTAGONISTS HAVING SUBSTITUTED (b)-AMINO ACID RESIDUES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME NIPPON STEEL CORP (JP) 2001-09-19 EP disclosed
US-5866592-A Fibrinogen receptor antagonist and pharmaceutical compositions comprising the same NIPPON STEEL CORPORATION (JP) 1999-02-02 US disclosed