SCHEMBL7835873

SCHEMBL7835873

CC(C)(NC(=O)c1ccc(C#N)cc1)C(C(=O)N1CCC(CC(=O)OCc2ccccc2)CC1)c1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
YAP1 P46937 2/20 0.41
CHRM4 P08173 4/20 0.41
KMT2A Q03164 1/20 0.41
EPHX2 P34913 1/20 0.39
CCR3 P51677 1/20 0.39
PRSS1 P07477 2/20 0.39
CTSG P08311 2/20 0.39
CTRB1 P17538 2/20 0.39
CMA1 P23946 2/20 0.39
KCNH2 Q12809 1/20 0.38
CCKBR P32239 1/20 0.37
KDM1A O60341 2/20 0.37
P2RX7 Q99572 1/20 0.37
CACNA1F O60840 1/20 0.37
HTR1A P08908 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
DRD2 P14416 1/20 0.37
CNR1 P21554 1/20 0.37
DRD1 P21728 1/20 0.37
DRD4 P21917 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7836339 0.94 YAP1 (0.44) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7357897 0.92 YAP1 (0.46) YAP1CHRM4KMT2ACCR3PRSS1
SCHEMBL7833217 0.91 GRIN2B (0.42) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7839324 0.89 ITGB3 (0.44) YAP1CHRM4KMT2ACCR3PRSS1
SCHEMBL7834829 0.88 ITGB3 (0.48) PRSS1
SCHEMBL7833800 0.86 YAP1 (0.44) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7836103 0.86 CTSG (0.43) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7833534 0.86 YAP1 (0.43) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7835452 0.84 PRSS1 (0.44) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7362435 0.83 ITGB3 (0.41) YAP1CHRM4CCKBRP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800516-B1 FIBRINOGEN RECEPTOR ANTAGONISTS HAVING SUBSTITUTED (b)-AMINO ACID RESIDUES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME NIPPON STEEL CORP (JP) 2001-09-19 EP disclosed
US-5866592-A Fibrinogen receptor antagonist and pharmaceutical compositions comprising the same NIPPON STEEL CORPORATION (JP) 1999-02-02 US disclosed