SCHEMBL7363405

SCHEMBL7363405

COC(=O)CC(C#N)c1ccc(OC)c(OC)c1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
KDM4E B2RXH2 1/20 0.54
LMNA P02545 1/20 0.54
MAPT P10636 1/20 0.54
HTT P42858 1/20 0.54
TNF P01375 9/20 0.52
PDE4A P27815 3/20 0.52
PDE4B Q07343 3/20 0.52
PDE4C Q08493 3/20 0.52
PDE4D Q08499 3/20 0.52
ACHE P22303 4/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C19 P33261 1/20 0.45
KMT2A Q03164 1/20 0.44
TSHR P16473 1/20 0.44
RAB9A P51151 1/20 0.44
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7294570 0.88 ALDH1A1 (0.54) ALDH1A1KDM4ELMNAMAPTHTT
SCHEMBL9155153 0.87 ALDH1A1 (0.55) ALDH1A1KDM4ELMNAMAPTHTT
SCHEMBL30530004 0.86 PDE4B (0.60) PDE4APDE4BPDE4CPDE4D
SCHEMBL7363289 0.86 PDE4B (0.60) PDE4APDE4BPDE4CPDE4D
SCHEMBL4683616 0.80 HTT (0.43) ALDH1A1LMNAMAPTHTTTNF
SCHEMBL7744741 0.80 KMT2A (0.47) ALDH1A1KDM4EMAPTHTTPDE4A
SCHEMBL30147220 0.80 ACHE (0.53) ALDH1A1KDM4ELMNAMAPTHTT
SCHEMBL7366317 0.79 PDE4A (0.53) PDE4APDE4BPDE4CPDE4D
SCHEMBL8771052 0.79 TNF (0.56) ALDH1A1TNFPDE4APDE4BPDE4C
SCHEMBL31467205 0.79 HTT (0.48) ALDH1A1KDM4ELMNAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0584208-A4 1994-03-23 EP disclosed
EP-0584208-A1 PYRROLIDINONES SMITHKLINE BEECHAM CORPORATION (US) 1994-03-02 EP disclosed
WO-1992019594-A1 PYRROLIDINONES SMITHKLINE BEECHAM CORPORATION (US) 1992-11-12 WO disclosed