SCHEMBL7744741

SCHEMBL7744741

COC(=O)CC(C#N)c1ccc(F)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.47
HTT P42858 2/20 0.41
MAPT P10636 6/20 0.41
ALDH1A1 P00352 2/20 0.41
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
MME P08473 1/20 0.37
FFAR1 O14842 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
GAA P10253 3/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RAB9A P51151 1/20 0.36
DPP4 P27487 2/20 0.36
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7831088 0.82 FFAR1 (0.49) KMT2ACES2CES1MMEFFAR1
SCHEMBL10634846 0.82 KMT2A (0.52) KMT2AHTTMAPTALDH1A1CES2
SCHEMBL30529996 0.81 L3MBTL1 (0.46) KMT2AHTTMAPTALDH1A1FFAR1
SCHEMBL7363405 0.80 ALDH1A1 (0.54) KMT2AHTTMAPTALDH1A1PDE4A
SCHEMBL4683616 0.80 HTT (0.43) KMT2AHTTMAPTALDH1A1RAB9A
SCHEMBL8770875 0.79 CES2 (0.45) KMT2AHTTMAPTALDH1A1CES2
SCHEMBL435332 0.79 ESR1 (0.51) KMT2AHTTMAPTALDH1A1MEN1
SCHEMBL20967754 0.79 CES2 (0.45) KMT2AHTTMAPTALDH1A1CES2
SCHEMBL30955364 0.79 CES2 (0.45) KMT2AHTTMAPTALDH1A1CES2
SCHEMBL31467205 0.79 HTT (0.48) KMT2AHTTMAPTALDH1A1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242607-B1 SUCH AS 4-CYANO-4-(3,4-DICHLOROPHENYL)HEPTANEDIOIC ACID USED AS ANTAGONISTS OF NEUROKININES SANOFI-SYNTHELABO (FR) 2001-06-05 US disclosed
US-6008360-A Substituted 3-aryl-3-carboxyalkyl glutaramides, method for preparing same by 4-arylo-4-cyanoheptane dicarboxylic acid cyclisation, and use thereof for preparing 3-aryl-3-hydroxyalkylpiperidines SANOFI-SYNTHELABO (FR) 1999-12-28 US disclosed