SCHEMBL7364733

SCHEMBL7364733

[CH]c1cccnc1Oc1cccc(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.47
LCK P06239 1/20 0.47
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
MEN1 O00255 1/20 0.45
PPP1CA P62136 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
P2RY1 P47900 2/20 0.42
CYP19A1 P11511 1/20 0.39
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
SCN5A Q14524 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1552831 0.81 PDE4A (0.46) EGFRLCKPDE4APDE4BPDE4C
SCHEMBL6136758 0.81 PDE4A (0.55) EGFRLCKPDE4APDE4BPDE4C
SCHEMBL27535812 0.78 KMT2A (0.58) EGFRLCKPDE4APDE4BPDE4C
SCHEMBL11373704 0.78 EGFR (0.47) EGFRLCKPDE4APDE4BPDE4C
SCHEMBL7370543 0.77 MEN1 (0.58) EGFRLCKPDE4APDE4BPDE4C
SCHEMBL7366622 0.77 ALDH1A1 (0.44) EGFRLCKPDE4APDE4BPDE4C
SCHEMBL7367307 0.77 AR (0.50) EGFRLCKPDE4APDE4BPDE4C
SCHEMBL7674124 0.76 ALDH1A1 (0.58) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL2332693 0.76 ALDH1A1 (0.61) ALDH1A1POLBGAAP2RY1RAB9A
SCHEMBL7364681 0.75 RAB9A (0.72) PDE4APDE4BPDE4CPDE4DALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0971894-A1 NICOTINAMIDE DERIVATIVES Pfizer Products Inc. (US) 2000-01-19 EP disclosed
WO-1998045268-A1 NICOTINAMIDE DERIVATIVES PFIZER PRODUCTS INC. (US) 1998-10-15 WO disclosed