SCHEMBL7365480

SCHEMBL7365480

CC(C)[C@H](NC(=O)[C@H](Cc1ccccc1F)NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 5/20 0.57
MME P08473 4/20 0.57
CTSB P07858 4/20 0.53
CTSK P43235 4/20 0.53
CTSL P07711 5/20 0.51
CTSS P25774 1/20 0.51
CASP3 P42574 1/20 0.50
TACR1 P25103 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275434 0.88 ECE1 (0.65) ECE1MMECTSBCTSKCTSL
SCHEMBL14438411 0.85 ITGB3 (0.56) ECE1MMECTSBCTSKCTSL
SCHEMBL7444291 0.85 ITGB3 (0.56) ECE1MMECTSBCTSKCTSL
SCHEMBL5561541 0.83 ALDH1A1 (0.60) CTSBCTSKCTSLCTSSTACR1
SCHEMBL5561531 0.83 ALDH1A1 (0.60) CTSBCTSKCTSLCTSSTACR1
SCHEMBL7355798 0.82 CTSK (0.74) CTSBCTSKCTSLCTSS
SCHEMBL7355802 0.82 CTSK (0.74) CTSBCTSKCTSLCTSS
SCHEMBL6150075 0.81 ECE1 (0.48) ECE1MMECTSBCTSKCTSL
SCHEMBL6272667 0.80 ECE1 (0.64) ECE1MMECTSBCTSKCTSL
SCHEMBL7378851 0.80 ECE1 (0.64) ECE1MMECTSBCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998025949-A1 SUBSTITUTED 5-AMINO-1,3,4-THIADIAZOLE-2-THIONES PROSCRIPT, INC. (US) 1998-06-18 WO disclosed
EP-0845002-A2 AMINO ACID AMIDES OF 5-AMINO-1,3,4-THIADIAZONES AND THEIR USE AS INHIBITORS FOR MATRIX METALLOPROTEINASES PROSCRIPT, INC. (US) 1998-06-03 EP disclosed
US-5677282-A ENZYME INHIBITOR; OSTEOARTHRITIS AND RHEUMATIC DISORDERS PROSCRIPT, INC. (US) 1997-10-14 US disclosed
WO-1996040745-A2 AMINO ACID AMIDES OF 5-AMINO-1,3,4-THIADIAZONES AND THEIR USE AS INHIBITORS FOR MATRIX METALLOPROTEINASES PROSCRIPT, INC. (US) 1996-12-19 WO disclosed