SCHEMBL7365563

SCHEMBL7365563

COC(=O)c1cccc(-c2oc(=O)c3ccc[nH]c2-3)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 1/20 0.46
DHODH Q02127 1/20 0.43
ERN1 O75460 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
MAPT P10636 1/20 0.43
BLM P54132 1/20 0.43
KMT2A Q03164 1/20 0.43
SAE1 Q9UBE0 1/20 0.43
UBA2 Q9UBT2 1/20 0.43
CA12 O43570 2/20 0.41
CA9 Q16790 2/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
PIK3CG P48736 1/20 0.41
PRKDC P78527 1/20 0.41
GPR119 Q8TDV5 1/20 0.41
PDK2 Q15119 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7365409 0.88 ALDH1A1 (0.44) NPC1RAB9AALDH1A1MAPTKMT2A
SCHEMBL7370381 0.83 NR4A2 (0.37) ALDH1A1GPR119
SCHEMBL7364705 0.82 CDK8 (0.46) CDK8ERN1ALDH1A1POLBMAPT
SCHEMBL7368565 0.81 ALDH1A1 (0.50) NPC1RAB9AALDH1A1MAPTKMT2A
SCHEMBL7365581 0.75 CDK8 (0.48) CDK8DHODHERN1NPC1RAB9A
SCHEMBL7366065 0.74 MIF (0.39) NPC1RAB9AALDH1A1KMT2ACA12
SCHEMBL7363528 0.73 IKBKB (0.40) NPC1RAB9AALDH1A1PRKDCPDPK1
SCHEMBL7363579 0.72 MAPT (0.49) ERN1ALDH1A1MAPTKMT2APDK2
SCHEMBL9950445 0.72 CDK8 (0.59) CDK8ERN1CA12CA9CA1
SCHEMBL7364846 0.72 NPC1 (0.43) NPC1RAB9AALDH1A1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716954-A ANTIINFLAMMATORY AGENT, ANTIHISTAMINES, IMMUNOSUPPRESSION,AUTOIMMUNE DISEASES SYNTEX U.S.A. INC. (US) 1998-02-10 US disclosed
EP-0612321-A1 PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1994-08-31 EP disclosed
WO-1993007146-A1 BENZO AND PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1993-04-15 WO disclosed