SCHEMBL7370381

SCHEMBL7370381

COC(=O)c1cc(-c2oc(=O)c3ccc[nH]c2-3)ccc1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 5/20 0.37
SLC6A3 Q01959 4/20 0.37
SLC6A4 P31645 3/20 0.37
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
SLC6A2 P23975 1/20 0.37
ROCK2 O75116 1/20 0.37
CSF1R P07333 1/20 0.37
KDR P35968 1/20 0.37
FLT3 P36888 1/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
CDK5 Q00535 1/20 0.37
ROCK1 Q13464 1/20 0.37
SLK Q9H2G2 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.37
TDP2 O95551 1/20 0.36
THRB P10828 1/20 0.36
ESR2 Q92731 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7365563 0.83 CDK8 (0.46) ALDH1A1GPR119
SCHEMBL7365409 0.83 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDATM
SCHEMBL7361974 0.76 NR4A2 (0.36) NR4A2SLC6A3SLC6A4SLC6A2ROCK2
SCHEMBL7364846 0.76 NPC1 (0.43) ALDH1A1KDM4EHPGDKDR
SCHEMBL7368721 0.75 KMT2A (0.43) ALDH1A1KDM4E
SCHEMBL7367312 0.75 ALDH1A1 (0.47) ALDH1A1KDM4EHPGD
SCHEMBL7368565 0.74 ALDH1A1 (0.50) ALDH1A1KDM4EHPGD
SCHEMBL7366065 0.72 MIF (0.39) ALDH1A1KDM4E
SCHEMBL70184 0.72 KDM4E (0.47) NR4A2SLC6A3SLC6A4ALDH1A1KDM4E
SCHEMBL7363528 0.71 IKBKB (0.40) ALDH1A1KDM4EHPGDCREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716954-A ANTIINFLAMMATORY AGENT, ANTIHISTAMINES, IMMUNOSUPPRESSION,AUTOIMMUNE DISEASES SYNTEX U.S.A. INC. (US) 1998-02-10 US disclosed
EP-0612321-A1 PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1994-08-31 EP disclosed
WO-1993007146-A1 BENZO AND PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1993-04-15 WO disclosed