SCHEMBL7365937

SCHEMBL7365937

CCCCOC(=O)NC(CC=O)C(=O)OCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSK P43235 10/20 0.54
CTSS P25774 4/20 0.52
CTSL P07711 3/20 0.52
ALDH1A1 P00352 1/20 0.51
CYP3A4 P08684 1/20 0.51
TSHR P16473 1/20 0.51
MAPK1 P28482 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
SIRT2 Q8IXJ6 2/20 0.46
SIRT1 Q96EB6 2/20 0.46
CTSB P07858 1/20 0.46
SIRT3 Q9NTG7 1/20 0.45
CAPN1 P07384 1/20 0.45
CAPN2 P17655 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL254236 0.95 CTSL (0.55) CTSKCTSSCTSLALDH1A1CYP3A4
SCHEMBL28190849 0.87 CTSL (0.54) CTSKCTSSCTSLALDH1A1CYP3A4
SCHEMBL3188496 0.87 CTSK (0.53) CTSKCTSSCTSLALDH1A1CTSB
SCHEMBL16862505 0.87 CTSK (0.53) CTSKCTSSCTSLALDH1A1CTSB
SCHEMBL7761583 0.86 CTSS (0.55) CTSKCTSSCTSLALDH1A1CYP3A4
SCHEMBL15569565 0.86 CTSS (0.55) CTSKCTSSCTSLALDH1A1CYP3A4
SCHEMBL5550159 0.86 CTSS (0.55) CTSKCTSSCTSLALDH1A1CYP3A4
SCHEMBL6254290 0.85 CASP1 (0.57) CTSKCTSSCTSLALDH1A1CYP3A4
SCHEMBL27617576 0.85 CTSS (0.54) CTSKCTSSCTSLALDH1A1CYP3A4
SCHEMBL4452037 0.85 CASP1 (0.57) CTSKCTSSCTSLALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1204652-A1 NOVEL SUCCINATE DERIVATIVE COMPOUNDS USEFUL AS CYSTEINE PROTEASE INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2002-05-15 EP disclosed
WO-2001009110-A1 NOVEL SUCCINATE DERIVATIVE COMPOUNDS USEFUL AS CYSTEINE PROTEASE INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-02-08 WO disclosed