SCHEMBL7366389

SCHEMBL7366389

CN1c2ccc(C(=O)O)cc2CNC(=O)[C@@H]1CC(=O)O

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.43
ALDH1A1 P00352 8/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
TDP1 Q9NUW8 1/20 0.38
ITGB3 P05106 2/20 0.38
ITGA2B P08514 1/20 0.38
KDM4E B2RXH2 2/20 0.37
POLB P06746 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.35
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
ITGAV P06756 1/20 0.35
MAPT P10636 1/20 0.35
HDAC2 Q92769 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7078805 1.00 TSHR (0.43) TSHRALDH1A1SMN1; SMN2L3MBTL1TDP1
SCHEMBL7333012 0.86 TSHR (0.39) TSHRALDH1A1SMN1; SMN2L3MBTL1TDP1
SCHEMBL7919242 0.85 TSHR (0.43) TSHRALDH1A1SMN1; SMN2L3MBTL1TDP1
SCHEMBL7401266 0.85 TSHR (0.43) TSHRALDH1A1SMN1; SMN2L3MBTL1TDP1
SCHEMBL7079518 0.83 TSHR (0.36) TSHRALDH1A1SMN1; SMN2L3MBTL1TDP1
SCHEMBL7658169 0.81 ITGB3 (0.56) TSHRALDH1A1SMN1; SMN2L3MBTL1TDP1
SCHEMBL7399769 0.81 HTT (0.45) TSHRALDH1A1TDP1POLBLMNA
SCHEMBL5155939 0.79 ITGB3 (0.41) ITGB3ITGA2BLMNAITGAVMAPT
SCHEMBL7368305 0.78 ITGB3 (0.60) ITGB3ITGA2BTP53ITGAVMAPT
SCHEMBL23535782 0.76 LMNA (0.49) ALDH1A1L3MBTL1TDP1KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0767792-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-11-20 EP disclosed
EP-0767792-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-04-16 EP disclosed
WO-1996000730-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1996-01-11 WO disclosed