SCHEMBL7367039

SCHEMBL7367039

COC(C=O)[C@H]1C(=O)N(OC(=O)COC(=O)C(F)(F)F)CCN1C(=O)C(N)CC(=O)N1CCN(c2ccncc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.39
DPP8 Q6V1X1 3/20 0.39
DPP7 Q9UHL4 3/20 0.39
CYP3A4 P08684 3/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
ITGB3 P05106 1/20 0.30
ITGA2B P08514 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7364293 0.87 DPP8 (0.41) DPP4DPP8DPP7CYP3A4CYP2D6
SCHEMBL7372151 0.85 DPP4 (0.40) DPP4DPP8DPP7CYP3A4CYP2D6
SCHEMBL7369431 0.75 L3MBTL1 (0.34) DPP4DPP8DPP7CYP3A4CYP2D6
SCHEMBL7367999 0.74 ALDH1A1 (0.39) ITGB3ITGA2BALDH1A1GAA
SCHEMBL7438854 0.72 DPP8 (0.42) DPP4DPP8DPP7CYP3A4CYP2D6
Trifluoroacetic Acid SCHEMBL7924834 0.71 DPP8 (0.47) DPP4DPP8DPP7CYP3A4CYP2D6
Trifluoroacetic Acid SCHEMBL7364289 0.71 DPP8 (0.47) DPP4DPP8DPP7CYP3A4CYP2D6
Trifluoroacetic Acid SCHEMBL7365694 0.71 DPP8 (0.47) DPP4DPP8DPP7CYP3A4CYP2D6
SCHEMBL7937529 0.67 RORC (0.35) ITGB3ITGA2BALDH1A1
SCHEMBL7372688 0.67 CASP1 (0.36) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970071-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 2000-01-12 EP disclosed
WO-1998039324-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-11 WO disclosed