SCHEMBL7367816

SCHEMBL7367816

CC(C)(C)OC(=O)CNC(=O)c1ccc2c(NC(N)=NCl)cncc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRC P08575 2/20 0.42
MAPT P10636 4/20 0.34
DGAT2 Q96PD7 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GABRA5 P31644 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
F2 P00734 2/20 0.33
HPGDS O60760 1/20 0.33
STAMBP O95630 1/20 0.32
F10 P00742 1/20 0.32
F7 P08709 1/20 0.32
F3 P13726 1/20 0.32
SIRT2 Q8IXJ6 1/20 0.32
SIRT1 Q96EB6 1/20 0.32
SIRT3 Q9NTG7 1/20 0.32
LATS1 O95835 1/20 0.32
CYP17A1 P05093 1/20 0.32
CYP3A4 P08684 1/20 0.32
NAMPT P43490 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7363404 0.92 DGAT2 (0.41) PTPRCMAPTDGAT2KMT2ACYP17A1
SCHEMBL7372152 0.85 AKT1 (0.32) MEN1KMT2AF2HPGDS
SCHEMBL7050306 0.82 PLAU (0.37) MAPTKDM4EF2
SCHEMBL7378246 0.80 CA1 (0.42) KDM4E
SCHEMBL6437619 0.79 PTPRC (0.42) PTPRCMAPTDGAT2KDM4EGABRA5
SCHEMBL7375649 0.78 NR1D1 (0.35) MAPTKDM4EMEN1KMT2A
SCHEMBL7050066 0.77 PLAU (0.39) MAPTMEN1KMT2ACYP3A4
SCHEMBL7368535 0.76 NR1D1 (0.35) KDM4E
SCHEMBL7370338 0.75 PLAU (0.34) F2F10
SCHEMBL7048344 0.74 PLAU (0.42) MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242120-A2 COMBINATIONS OF GROWTH FACTORS AND I:UPA OR I:MMP FOR THE TREATMENT OF DAMAGED TISSUE Pfizer Limited (GB) 2002-09-25 EP disclosed
WO-2001049309-A2 COMBINATIONS OF GROWTH FACTORS AND I: UPA OR I: MMP FOR THE TREATMENT OF DAMAGED TISSUE PFIZER LIMITED (GB) 2001-07-12 WO disclosed
EP-1077945-A1 ISOQUINOLINES AS UROKINASE INHIBITORS PFIZER INC. (US) 2001-02-28 EP disclosed
WO-2000005214-A2 ISOQUINOLINES AS UROKINASE INHIBITORS PFIZER INC. (US) 2000-02-03 WO disclosed