SCHEMBL7368434

SCHEMBL7368434

Cc1ccc(-c2ccccc2C(=O)Nc2ccc(C(=O)N(C)c3ccccc3C)cc2C)cc1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.52
GAA P10253 1/20 0.47
MTTP P55157 5/20 0.46
HSD17B1 P14061 1/20 0.44
HSD17B2 P37059 1/20 0.44
MAPT P10636 2/20 0.43
PKM P14618 1/20 0.43
LMNA P02545 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
F10 P00742 1/20 0.41
KLK1 P06870 1/20 0.41
KLK5 Q9Y337 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7378000 0.89 ALDH1A1 (0.51) ALDH1A1GAAMTTPMAPTLMNA
SCHEMBL7376741 0.87 CHRNB2 (0.49) ALDH1A1GAAHSD17B1HSD17B2LMNA
SCHEMBL7373393 0.86 ALDH1A1 (0.47) ALDH1A1GAAMTTPMAPTF10
SCHEMBL7376100 0.84 ALDH1A1 (0.43) ALDH1A1GAAMTTPMAPTL3MBTL1
SCHEMBL7376852 0.82 F10 (0.48) ALDH1A1GAAMTTPHSD17B1HSD17B2
SCHEMBL7748399 0.81 ALDH1A1 (0.51) ALDH1A1GAAMTTPMAPTLMNA
SCHEMBL7372810 0.81 ALDH1A1 (0.44) ALDH1A1MTTPMAPTL3MBTL1
SCHEMBL7376652 0.79 PTGER1 (0.46) ALDH1A1MTTPMAPTL3MBTL1F10
SCHEMBL7375925 0.79 MTTP (0.40) ALDH1A1GAAMTTPMAPT
SCHEMBL7513968 0.79 RAB9A (0.46) ALDH1A1GAAMAPTLMNAF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211242-B1 CARDIOVASCULAR DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
EP-0757670-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 1999-01-13 EP disclosed
WO-1995029152-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-02 WO disclosed