SCHEMBL7373393

SCHEMBL7373393

Cc1ccc(-c2ccccc2C(=O)Nc2ccc(C(=O)N(C)c3ccc(Cl)cc3O)cc2C)cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
F10 P00742 4/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KCNMA1 Q12791 1/20 0.44
MTTP P55157 3/20 0.43
MAPT P10636 1/20 0.42
SERPINE1 P05121 1/20 0.41
KLK1 P06870 1/20 0.41
KLK5 Q9Y337 1/20 0.41
TP53 P04637 1/20 0.41
AVPR2 P30518 1/20 0.41
AVPR1A P37288 1/20 0.41
GAA P10253 2/20 0.41
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
TAS1R2 Q8TE23 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7513968 0.93 RAB9A (0.46) ALDH1A1F10NPC1RAB9AKCNMA1
SCHEMBL8812136 0.90 SMN1; SMN2 (0.46) ALDH1A1F10NPC1RAB9ASMN1; SMN2
SCHEMBL7371628 0.89 KCNMA1 (0.48) ALDH1A1F10NPC1RAB9ASMN1; SMN2
SCHEMBL7376165 0.89 AVPR2 (0.48) ALDH1A1F10NPC1RAB9ASMN1; SMN2
SCHEMBL7368434 0.86 ALDH1A1 (0.52) ALDH1A1F10MTTPMAPTKLK1
SCHEMBL7376652 0.85 PTGER1 (0.46) ALDH1A1F10NPC1RAB9ASMN1; SMN2
SCHEMBL7377166 0.82 AVPR2 (0.48) NPC1RAB9ASMN1; SMN2MAPTTP53
SCHEMBL7512858 0.81 ALDH1A1 (0.50) ALDH1A1NPC1RAB9ASMN1; SMN2KCNMA1
SCHEMBL7376778 0.80 NPC1 (0.51) F10NPC1RAB9ASMN1; SMN2TP53
SCHEMBL8813752 0.80 KCNMA1 (0.49) ALDH1A1F10NPC1SMN1; SMN2KCNMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211242-B1 CARDIOVASCULAR DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
WO-1995029152-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-02 WO disclosed