SCHEMBL7368442

SCHEMBL7368442

CCC(CCCc1ccccc1)c1cc(O)c(C(c2cccc(NS(=O)(=O)c3ccccc3)c2)C2CC2)c(=O)o1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 5/20 0.39
MAP1LC3B Q9GZQ8 1/20 0.38
MAP1LC3A Q9H492 1/20 0.38
PTGES O14684 1/20 0.38
HDAC8 Q9BY41 2/20 0.35
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
OPRM1 P35372 2/20 0.35
F2 P00734 1/20 0.34
F10 P00742 1/20 0.34
PRSS1 P07477 1/20 0.34
HDAC1 Q13547 2/20 0.34
LIMK1 P53667 1/20 0.34
LIMK2 P53671 1/20 0.34
MLNR O43193 1/20 0.34
NR1I2 O75469 1/20 0.34
ABCB11 O95342 1/20 0.34
PGR P06401 1/20 0.34
CTSD P07339 1/20 0.34
CHRM2 P08172 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6173713 0.91 PTGES (0.38) HTR6MAP1LC3BMAP1LC3APTGESHDAC1
SCHEMBL7443310 0.89 POLB (0.36) HTR6MAP1LC3BMAP1LC3APTGESCTSD
SCHEMBL7371939 0.88 HTR6 (0.41) HTR6MAP1LC3BMAP1LC3APTGESHDAC8
SCHEMBL6174303 0.86 ITGA1 (0.40) PTGESHDAC1LIMK1LIMK2CTSD
SCHEMBL7482607 0.86 ALDH1A1 (0.40) MAP1LC3BMAP1LC3ALIMK1LIMK2LMNA
SCHEMBL6175248 0.86 CYP2C9 (0.38) HTR2B
SCHEMBL7440371 0.85 HDAC1 (0.37) HTR6MAP1LC3BMAP1LC3APTGESHDAC1
SCHEMBL7447436 0.85 LIMK2 (0.37) LIMK2
SCHEMBL6172890 0.85 LIMK2 (0.39) HDAC8HDAC1LIMK1LIMK2LMNA
SCHEMBL7441470 0.85 HTR6 (0.40) HTR6MAP1LC3BMAP1LC3APTGESHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729465-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP claimed
WO-1995014013-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO claimed