SCHEMBL7440371

SCHEMBL7440371

CCC(Cc1ccccc1)c1cc(O)c(C(c2cccc(NS(=O)(=O)c3ccc(NO)cc3)c2)C2CC2)c(=O)o1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.37
ALOX12 P18054 2/20 0.35
NAMPT P43490 1/20 0.35
MAP1LC3B Q9GZQ8 2/20 0.35
MAP1LC3A Q9H492 2/20 0.35
GPR27 Q9NS67 1/20 0.34
PTGES O14684 1/20 0.34
ALDH1A1 P00352 3/20 0.34
LIMK2 P53671 2/20 0.34
LIMK1 P53667 1/20 0.34
CTSD P07339 1/20 0.34
BACE1 P56817 1/20 0.34
BACE2 Q9Y5Z0 1/20 0.34
PDE4A P27815 1/20 0.33
SLC2A1 P11166 1/20 0.33
HTR6 P50406 2/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PTGIR P43119 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6173713 0.95 PTGES (0.38) HDAC1ALOX12NAMPTMAP1LC3BMAP1LC3A
SCHEMBL6174303 0.93 ITGA1 (0.40) HDAC1ALOX12GPR27PTGESLIMK2
SCHEMBL7482607 0.93 ALDH1A1 (0.40) MAP1LC3BMAP1LC3AALDH1A1LIMK2LIMK1
SCHEMBL7447436 0.92 LIMK2 (0.37) ALOX12LIMK2
SCHEMBL6172890 0.92 LIMK2 (0.39) HDAC1ALDH1A1LIMK2LIMK1
SCHEMBL7439445 0.91 LIMK2 (0.36) NAMPTMAP1LC3BMAP1LC3APTGESALDH1A1
SCHEMBL6176577 0.91 IKBKB (0.44) ALDH1A1SMN1; SMN2
SCHEMBL6175855 0.91 CYP19A1 (0.41) ALOX12GPR27ALDH1A1LIMK2HTT
SCHEMBL6174297 0.90 PGAM1 (0.38) GPR27PTGIR
SCHEMBL7402228 0.90 KDM1A (0.39) HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed