SCHEMBL7374140

SCHEMBL7374140

Cc1cccc(N(C)C(=O)c2ccc(N)cc2)c1

nearest known ligand 0.71

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 12/20 0.71
HSD17B2 P37059 12/20 0.71
SIGMAR1 Q99720 1/20 0.47
KDM4E B2RXH2 2/20 0.46
LMNA P02545 1/20 0.46
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HSD17B10 Q99714 1/20 0.46
THRB P10828 1/20 0.44
NPC1 O15118 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21241029 0.89 HSD17B1 (0.83) HSD17B1HSD17B2KDM4ELMNATSHR
SCHEMBL18585406 0.87 HSD17B1 (0.53) HSD17B1HSD17B2KDM4ELMNAHTT
SCHEMBL29940968 0.85 HSD17B2 (0.72) HSD17B1HSD17B2KDM4ELMNATSHR
SCHEMBL10212283 0.85 HSD17B2 (0.72) HSD17B1HSD17B2KDM4ELMNATSHR
SCHEMBL21620298 0.84 HSD17B1 (0.71) HSD17B1HSD17B2LMNANPC1
SCHEMBL94811 0.84 HSD17B1 (0.71) HSD17B1HSD17B2SIGMAR1KDM4ELMNA
SCHEMBL7368760 0.83 HTR3E (0.54) HSD17B1HSD17B2KDM4ESMN1; SMN2NPC1
SCHEMBL4658072 0.82 HSD17B1 (0.68) HSD17B1HSD17B2HTT
SCHEMBL7373511 0.82 KMT2A (0.64) KDM4ENPC1HTT
SCHEMBL7376609 0.81 HSD17B2 (0.75) HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211242-B1 CARDIOVASCULAR DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
EP-0757670-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 1999-01-13 EP disclosed
EP-0757670-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-12 EP disclosed
WO-1995029152-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-02 WO disclosed