SCHEMBL7368901

SCHEMBL7368901

CC(C)C(=O)Nc1nc(-c2cc(CC(C)C(=O)O)c(CC(C)C(=O)O)c([N+](=O)[O-])c2)cs1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.56
MAPT P10636 8/20 0.43
KMT2A Q03164 8/20 0.43
MEN1 O00255 7/20 0.43
ALDH1A1 P00352 4/20 0.43
HTT P42858 2/20 0.43
TYR P14679 1/20 0.43
RAB9A P51151 4/20 0.41
ATM Q13315 1/20 0.40
TP53 P04637 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
THRB P10828 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
MITF O75030 1/20 0.39
NTSR1 P30989 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8731806 0.76 LMNA (0.57) LMNAMAPTKMT2AMEN1ALDH1A1
SCHEMBL7372881 0.75 TP53 (0.37) MAPTTP53
SCHEMBL7372642 0.73 CES2 (0.30) LMNAALDH1A1HTTSMN1; SMN2CYP1A2
SCHEMBL7367277 0.70 MET (0.40) LMNAMAPTALDH1A1RAB9AATM
SCHEMBL2752589 0.69 LMNA (0.68) LMNAMAPTKMT2AMEN1ALDH1A1
SCHEMBL7373077 0.66 MEN1 (0.39) KMT2AMEN1
SCHEMBL9891792 0.65 ABL1 (0.72) LMNAMAPTKMT2AMEN1ALDH1A1
SCHEMBL9891898 0.65 LMNA (0.69) LMNAMAPTKMT2AMEN1ALDH1A1
SCHEMBL7369806 0.64 KMT2A (0.42) LMNAMAPTKMT2AMEN1ALDH1A1
SCHEMBL18424368 0.63 ABL1 (0.67) LMNAMAPTKMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0237929-B1 3,5-DISUBSTITUTED PYROCATECHOL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-06-02 EP disclosed
EP-0237929-A1 3,5-Disubstituted pyrocatechol derivatives F. HOFFMANN-LA ROCHE AG (CH) 1987-09-23 EP disclosed