SCHEMBL7369546

SCHEMBL7369546

O=C(CC1Oc2ccc(C[C@H](NS(=O)(=O)c3ccccc3)C(=O)OCc3ccccc3)cc2NC1=O)Nc1ncc[nH]1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.39
HSD17B10 Q99714 3/20 0.38
TSHR P16473 2/20 0.38
MAPT P10636 2/20 0.38
KMT2A Q03164 6/20 0.37
MEN1 O00255 5/20 0.37
MAPK1 P28482 2/20 0.37
ALOX15 P16050 1/20 0.37
HTT P42858 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CTSL P07711 1/20 0.36
CTSS P25774 1/20 0.36
TP53 P04637 1/20 0.36
ALDH1A1 P00352 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGAV P06756 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7365336 0.95 TSHR (0.43) THRBHSD17B10TSHRMAPTKMT2A
SCHEMBL7468966 0.93 BDKRB1 (0.39) THRBHSD17B10TSHRMAPTKMT2A
SCHEMBL7163732 0.92 TSHR (0.41) THRBHSD17B10TSHRMAPTKMT2A
SCHEMBL7472452 0.92 THRB (0.39) THRBHSD17B10TSHRMAPTKMT2A
SCHEMBL7368383 0.89 GAA (0.37) THRBHSD17B10TSHRMAPTKMT2A
SCHEMBL7478535 0.89 THRB (0.40) THRBHSD17B10TSHRMAPTKMT2A
SCHEMBL7474158 0.88 ITGB3 (0.48) THRBHSD17B10TSHRKMT2AMEN1
SCHEMBL7368163 0.86 BACE1 (0.39) THRBHSD17B10TSHRMAPTMAPK1
SCHEMBL7365578 0.86 THRB (0.42) THRBHSD17B10TSHRMAPTKMT2A
SCHEMBL7364282 0.86 ALOX15 (0.41) THRBHSD17B10MAPK1ALOX15HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0964856-B1 BICYCLIC AMINO ACIDS MERCK PATENT GMBH (DE) 2002-10-09 EP disclosed
EP-0964856-A1 BICYCLIC AMINO ACIDS MERCK PATENT GmbH (DE) 1999-12-22 EP disclosed
WO-1998035949-A1 BICYCLIC AMINO ACIDS MERCK PATENT GMBH (DE) 1998-08-20 WO disclosed