SCHEMBL7370511

SCHEMBL7370511

Nc1nc(-c2ccc(N3CCOCC3)nc2)cs1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADK P55263 1/20 0.57
CNR2 P34972 6/20 0.51
ATR Q13535 3/20 0.51
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
MAPK1 P28482 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
MEN1 O00255 1/20 0.48
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48
KMT2A Q03164 1/20 0.48
AR P10275 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL129802 0.81 ALOX5 (0.57) NPC1RAB9AMAPK1SMN1; SMN2MEN1
SCHEMBL28528175 0.81 ADK (0.47) ADKCNR2ATR
SCHEMBL21495017 0.79 AR (0.50) NPC1RAB9AMAPK1SMN1; SMN2MEN1
SCHEMBL24170032 0.77 AR (0.48) ADKNPC1RAB9ASMN1; SMN2MEN1
SCHEMBL19899542 0.76 SMN1; SMN2 (0.54) NPC1RAB9ASMN1; SMN2MEN1LMNA
SCHEMBL29654073 0.76 CYP1A1 (0.61) NPC1RAB9AMAPK1SMN1; SMN2MEN1
SCHEMBL13815773 0.75 CNR2 (0.53) ADKCNR2ATR
SCHEMBL7294070 0.74 CNR2 (0.62) CNR2SMN1; SMN2MEN1LMNAMAPT
SCHEMBL17407205 0.74 RAB9A (0.49) NPC1RAB9AMAPK1SMN1; SMN2MEN1
SCHEMBL12293461 0.74 RAB9A (0.52) NPC1RAB9AMAPK1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11584742-B2 Substituted aminothiazoles as inhibitors of nucleases MASARYKOVA UNIVERZITA (CZ) 2023-02-21 US disclosed
US-20220002282-A1 SUBSTITUTED AMINOTHIAZOLES AS INHIBITORS OF NUCLEASES MASARYKOVA UNIVERZITA (CZ) 2022-01-06 US disclosed
CN-112313229-A Substituted aminothiazoles as inhibitors of nucleases 马萨里克大学 2021-02-02 CN disclosed
WO-2019201865-A1 SUBSTITUTED AMINOTHIAZOLES AS INHIBITORS OF NUCLEASES MASARYKOVA UNIVERZITA (CZ) 2019-10-24 WO disclosed
WO-2019201865-A1 SUBSTITUTED AMINOTHIAZOLES AS INHIBITORS OF NUCLEASES MASARYKOVA UNIVERZITA (CZ) 2019-10-24 WO disclosed
US-20020177594-A1 Inhibitors of histone deacetylase ABBOTT LABORATORIES 2002-11-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11584742-B2 Substituted aminothiazoles as inhibitors of nucleases RNASEH1, DNASE1, FEN1 ADK 1481/4885CNR2 4825/4885ATR 605/4885
US-20020177594-A1 Inhibitors of histone deacetylase HDAC1, HDAC11, HDAC3 ADK 3710/4885CNR2 4785/4885ATR 2981/4885
US-20220002282-A1 SUBSTITUTED AMINOTHIAZOLES AS INHIBITORS OF NUCLEASES RNASEH1, DNASE1, FEN1 ADK 1481/4885CNR2 4825/4885ATR 605/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.