SCHEMBL7370531

SCHEMBL7370531

NC(Cc1ccc(OCc2ccccc2)cc1)C(=O)NCCCn1ccnc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QPCT Q16769 2/20 0.66
ALDH1A1 P00352 1/20 0.57
HPGD P15428 1/20 0.57
DUSP3 P51452 1/20 0.57
PTPN5 P54829 1/20 0.57
PTPN11 Q06124 1/20 0.57
HMOX1 P09601 1/20 0.56
IDE P14735 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
CYP19A1 P11511 1/20 0.53
CYP11B1 P15538 1/20 0.53
CYP11B2 P19099 1/20 0.53
HRH4 Q9H3N8 1/20 0.51
PKM P14618 1/20 0.50
ADAMTS5 Q9UNA0 1/20 0.50
GAA P10253 3/20 0.49
REN P00797 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.48
CTSS P25774 1/20 0.48
CTSK P43235 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339691 0.86 CTSS (0.56) QPCTALDH1A1HPGDDUSP3PTPN5
SCHEMBL7369227 0.85 QPCT (0.63) QPCTALDH1A1HPGDDUSP3PTPN5
SCHEMBL7868636 0.82 PKM (0.73) QPCTALDH1A1HPGDHMOX1SMN1; SMN2
SCHEMBL7339684 0.80 QPCT (0.51) QPCTALDH1A1HPGDDUSP3PTPN5
SCHEMBL7404871 0.80 CTSS (0.55) QPCTALDH1A1HPGDDUSP3PTPN5
SCHEMBL8191918 0.77 TACR2 (0.51) ALDH1A1SMN1; SMN2GAAREN
SCHEMBL7371156 0.76 HTT (0.57) ALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL8189087 0.76 TDP1 (0.55) ALDH1A1SMN1; SMN2REN
SCHEMBL5759785 0.76 HMOX1 (0.85) QPCTHMOX1CYP19A1CYP11B1CYP11B2
SCHEMBL7698099 0.76 LNPEP (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US claimed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO claimed
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US disclosed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed