SCHEMBL7370913

SCHEMBL7370913

COc1ccc(-c2nc(-c3cccnc3)c(C)[nH]2)c(OC)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 5/20 0.57
CYP3A4 P08684 3/20 0.56
CYP1A1 P04798 2/20 0.56
CYP1A2 P05177 2/20 0.56
CYP1B1 Q16678 2/20 0.56
PDE2A O00408 1/20 0.53
CYP11B2 P19099 6/20 0.51
CYP11B1 P15538 5/20 0.51
CYP17A1 P05093 4/20 0.51
CYP19A1 P11511 1/20 0.49
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
HSD17B10 Q99714 1/20 0.46
SMPD3 Q9NY59 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
CYP2E1 P05181 1/20 0.45
CYP2C8 P10632 1/20 0.45
CYP2D6 P10635 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7365692 0.91 NPY5R (0.57) NPY5RCYP3A4CYP1A1CYP1A2CYP1B1
SCHEMBL7369602 0.87 NPY5R (0.56) NPY5RCYP3A4CYP1A1CYP1A2CYP1B1
SCHEMBL7372225 0.87 NPY5R (0.62) NPY5RCYP3A4CYP1A1CYP1A2CYP1B1
SCHEMBL7369909 0.85 NPC1 (0.52) NPY5RPDE2ASMPD3NPC1RAB9A
SCHEMBL7371445 0.85 NPY5R (0.67) NPY5RALDH1A1SMPD3
SCHEMBL7377111 0.85 NPY5R (0.54) NPY5RCYP3A4CYP1A1CYP1A2CYP1B1
SCHEMBL7369293 0.84 CYP3A4 (0.52) NPY5RCYP3A4CYP1A1CYP1A2CYP1B1
SCHEMBL7371561 0.84 PDE2A (0.56) NPY5RCYP3A4CYP1A1CYP1A2CYP1B1
SCHEMBL27674585 0.83 NPY5R (0.67) NPY5RCYP3A4CYP1A2CYP11B2CYP11B1
Hydrochloric Acid SCHEMBL7370882 0.83 PDE2A (0.55) NPY5RCYP3A4CYP1A1CYP1A2CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4822805-A ANTIINFLAMMATORY AGENTS, CARDIOTONIC AGENTS, ANTIPLATELET AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1989-04-18 US disclosed
CN-87105680-A Imidazolium compounds and preparation method thereof and comprise the pharmaceutical composition of this compound 1988-04-27 CN disclosed
EP-0257897-A1 Imidazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-03-02 EP disclosed