SCHEMBL7369293

SCHEMBL7369293

COc1ccc(-c2nc(-c3cccnc3)c(CO)[nH]2)c(OC)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.52
CYP1A2 P05177 2/20 0.52
CYP1A1 P04798 1/20 0.52
CYP1B1 Q16678 1/20 0.52
CYP11B2 P19099 9/20 0.50
CYP11B1 P15538 8/20 0.50
CYP17A1 P05093 4/20 0.50
PDE2A O00408 1/20 0.49
NPY5R Q15761 2/20 0.47
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CYP19A1 P11511 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
MKNK1 Q9BUB5 1/20 0.43
MKNK2 Q9HBH9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7372964 0.87 MKNK1 (0.41) CYP3A4CYP1A2CYP1A1CYP1B1CYP11B2
SCHEMBL7370913 0.84 NPY5R (0.57) CYP3A4CYP1A2CYP1A1CYP1B1CYP11B2
SCHEMBL7371561 0.78 PDE2A (0.56) CYP3A4CYP1A2CYP1A1CYP1B1CYP11B2
SCHEMBL7371766 0.77 PDE2A (0.53) CYP3A4CYP1A2CYP1A1CYP1B1CYP11B2
Hydrochloric Acid SCHEMBL7370882 0.77 PDE2A (0.55) CYP3A4CYP1A2CYP1A1CYP1B1CYP11B2
SCHEMBL7365842 0.77 TGFBR1 (0.70) PDE2ANPY5RNPC1
SCHEMBL7365692 0.76 NPY5R (0.57) CYP3A4CYP1A2CYP1A1CYP1B1CYP11B2
SCHEMBL7369602 0.73 NPY5R (0.56) CYP3A4CYP1A2CYP1A1CYP1B1CYP11B2
SCHEMBL7372225 0.73 NPY5R (0.62) CYP3A4CYP1A2CYP1A1CYP1B1CYP11B2
SCHEMBL2817926 0.72 CYP11B1 (0.49) CYP11B1NPY5RKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4822805-A ANTIINFLAMMATORY AGENTS, CARDIOTONIC AGENTS, ANTIPLATELET AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1989-04-18 US disclosed
CN-87105680-A Imidazolium compounds and preparation method thereof and comprise the pharmaceutical composition of this compound 1988-04-27 CN disclosed
EP-0257897-A1 Imidazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-03-02 EP disclosed