SCHEMBL8177114

SCHEMBL8177114

O=C(NC(CNC(=O)c1nnc(CCCCNc2ccccn2)s1)C(=O)O)OCc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 14/20 0.61
ITGA2B P08514 5/20 0.61
ITGAV P06756 13/20 0.57
ITGB1 P05556 2/20 0.44
ITGA5 P08648 2/20 0.44
ANPEP P15144 1/20 0.43
GLS O94925 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8177121 1.00 ITGB3 (0.61) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7371601 0.85 ITGB3 (0.51) ITGB3ITGA2BITGAVGLS
SCHEMBL7371595 0.85 ITGB3 (0.51) ITGB3ITGA2BITGAVGLS
SCHEMBL8177327 0.84 ITGB3 (0.60) ITGB3ITGA2BITGAV
SCHEMBL7368311 0.83 ANPEP (0.45) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL8177321 0.79 ITGB3 (0.42) ITGB3ITGA2BITGAVGLS
SCHEMBL7368318 0.78 GLS (0.42) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7368315 0.78 GLS (0.42) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL8168274 0.77 ITGB3 (0.63) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL8179651 0.77 ITGAV (0.63) ITGB3ITGA2BITGAVITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153628-A 1,3,4-thiadiazoles and 1,3,4-Oxadiazoles as αv β3 antagonists DUPONT PHARMACEUTICALS COMPANY (US) 2000-11-28 US claimed
US-6153628-A 1,3,4-thiadiazoles and 1,3,4-Oxadiazoles as αv β3 antagonists DUPONT PHARMACEUTICALS COMPANY (US) 2000-11-28 US disclosed