SCHEMBL7373328

SCHEMBL7373328

NC[C](N)Cc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.48
CES2 O00748 1/20 0.48
AKR1B1 P15121 1/20 0.48
LOXL2 Q9Y4K0 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.44
CYP2A6 P11509 1/20 0.44
HTR2A P28223 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
HIF1A Q16665 1/20 0.44
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
HTT P42858 1/20 0.42
TSHR P16473 1/20 0.42
IDO1 P14902 3/20 0.41
NOS2 P35228 2/20 0.41
MEN1 O00255 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28085046 0.81 CES1 (0.55) CES1CES2AKR1B1LOXL2SMN1; SMN2
SCHEMBL8778515 0.78 CES2 (0.46) CES1CES2AKR1B1LOXL2SMN1; SMN2
SCHEMBL11795977 0.76 CES2 (0.44) CES1CES2AKR1B1LOXL2SMN1; SMN2
SCHEMBL8993215 0.76 CES1 (0.55) CES1CES2AKR1B1LOXL2SMN1; SMN2
SCHEMBL5184996 0.76 CES1 (0.55) CES1CES2AKR1B1LOXL2SMN1; SMN2
Phenylacetic Acid SCHEMBL28668840 0.73 AKR1B1 (0.81) CES1CES2AKR1B1HIF1AKMT2A
SCHEMBL1545179 0.73 CES1 (0.58) CES1CES2AKR1B1LOXL2HIF1A
SCHEMBL28045886 0.73 CES1 (0.46) CES1CES2AKR1B1LOXL2SMN1; SMN2
SCHEMBL9520947 0.73 ALDH1A1 (0.46) CES1CES2AKR1B1TAAR1HIF1A
SCHEMBL9701924 0.73 LOXL2 (0.43) CES1CES2AKR1B1LOXL2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722436-A4 MERCAPTOSULFIDE METALLOPROTEINASE INHIBITORS UNIV FLORIDA STATE (US) 1996-11-20 EP disclosed
EP-0722436-A1 MERCAPTOSULFIDE METALLOPROTEINASE INHIBITORS FLORIDA STATE UNIVERSITY (US) 1996-07-24 EP disclosed
WO-1995009833-A1 MERCAPTOSULFIDE METALLOPROTEINASE INHIBITORS FLORIDA STATE UNIVERSITY (US) 1995-04-13 WO disclosed