SCHEMBL9701924

SCHEMBL9701924

C=C=C(CN)Cc1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 2/20 0.43
HTR2A P28223 2/20 0.43
CYP2A6 P11509 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
AKR1B1 P15121 1/20 0.41
EPHX1 P07099 1/20 0.41
MAOA P21397 1/20 0.39
MMP2 P08253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11493475 0.98 LOXL2 (0.41) LOXL2HTR2ACYP2A6SMN1; SMN2TAAR1
SCHEMBL9702029 0.82 TAAR1 (0.48) TAAR1
SCHEMBL12003573 0.81 CES1 (0.43) CES2CES1AKR1B1EPHX1
SCHEMBL9700891 0.80 HTR2A (0.50) LOXL2HTR2ACYP2A6SMN1; SMN2TAAR1
SCHEMBL9701625 0.80 DRD2 (0.55) TAAR1
Hydrochloric Acid SCHEMBL9703374 0.79 KEAP1 (0.48) LOXL2HTR2ACYP2A6SMN1; SMN2TAAR1
SCHEMBL29029168 0.76 MEN1 (0.39) CES2CES1AKR1B1
SCHEMBL9701935 0.76 TAAR1 (0.52) SMN1; SMN2TAAR1
Hydrochloric Acid SCHEMBL9701893 0.76 MAOA (0.50) LOXL2HTR2ACYP2A6SMN1; SMN2TAAR1
SCHEMBL9701903 0.75 TAAR1 (0.52) TAAR1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120764-A Administering penicillamine and allenylamines to inhibit crosslinking of collagen MERRELL DOW PHARMACEUTICALS INC. (US) 1992-06-09 US disclosed
EP-0374440-A2 Inhibitors of lysyl oxidase MERRELL DOW PHARMACEUTICALS INC. (US) 1990-06-27 EP disclosed
EP-0011608-A1 Novel allenic amine and acid addition salts thereof, a process for their preparation, pharmaceutical preparations comprising them and the use of these compounds in the preparation of pharmaceutical compositions Astra Läkemedel Aktiebolag (SE) 1980-05-28 EP disclosed