SCHEMBL7375593

SCHEMBL7375593

COC(=O)N(NC(=O)c1cccc(NC(=N)N)c1)C(Cc1ccccc1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
RAB9A P51151 3/20 0.40
LMNA P02545 1/20 0.39
PARP1 P09874 1/20 0.39
PARP10 Q53GL7 1/20 0.39
NR1H4 Q96RI1 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CASR P41180 1/20 0.38
MAPT P10636 1/20 0.38
F2 P00734 1/20 0.38
F10 P00742 1/20 0.38
PRSS1 P07477 1/20 0.38
KCNK3 O14649 1/20 0.38
KCNK9 Q9NPC2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7409600 0.92 MAPT (0.42) ALDH1A1RAB9ALMNANR1H4MEN1
SCHEMBL7466483 0.92 NPC1 (0.45) ALDH1A1ITGB3ITGA2BRAB9ANR1H4
SCHEMBL7410381 0.91 ITGB3 (0.41) ITGB3ITGA2BLMNANR1H4MEN1
SCHEMBL7410551 0.91 ITGB3 (0.41) ITGB3ITGA2BLMNANR1H4MEN1
SCHEMBL7382269 0.90 NR1H4 (0.41) ALDH1A1ITGB3ITGA2BRAB9ALMNA
SCHEMBL7380572 0.89 ITGB3 (0.40) ALDH1A1ITGB3ITGA2BRAB9ALMNA
Phenylalanine SCHEMBL7414620 0.87 SLC7A5 (0.47) ALDH1A1ITGB3ITGA2BRAB9ASMN1; SMN2
SCHEMBL7382733 0.86 ALDH1A1 (0.45) ALDH1A1RAB9ALMNANR1H4MEN1
SCHEMBL7376793 0.86 RAB9A (0.38) ALDH1A1HPGDITGB3ITGA2BRAB9A
SCHEMBL7375609 0.85 ALDH1A1 (0.39) ALDH1A1HPGDITGB3ITGA2BRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP claimed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed