Phenylalanine

Phenylalanine

SCHEMBL7414620

CC(C)(C)OC(=O)N(NC(=O)c1cccc(NC(=N)N)c1)[C@@H](Cc1ccccc1)C(=O)O.N[C@@H](Cc1ccccc1)C(=O)O

nearest known ligand 0.47

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 5/20 0.47
NOS3 P29474 1/20 0.42
NOS1 P29475 1/20 0.42
NOS2 P35228 1/20 0.42
ITGB3 P05106 2/20 0.41
ITGAV P06756 2/20 0.41
ITGA2B P08514 2/20 0.41
ITGB1 P05556 1/20 0.39
ITGB5 P18084 1/20 0.39
BACE1 P56817 1/20 0.38
ALPI P09923 1/20 0.37
PKM P14618 1/20 0.37
PTGS1 P23219 1/20 0.37
XIAP P98170 1/20 0.37
CASR P41180 2/20 0.37
F2 P00734 4/20 0.36
TMPRSS6 Q8IU80 2/20 0.36
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TPH1 P17752 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7410551 0.96 ITGB3 (0.41) SLC7A5ITGB3ITGAVITGA2BITGB1
SCHEMBL7410381 0.96 ITGB3 (0.41) SLC7A5ITGB3ITGAVITGA2BITGB1
SCHEMBL7408424 0.87 ALDH1A1 (0.41) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL7375593 0.87 ALDH1A1 (0.42) ITGB3ITGA2BCASRF2ALDH1A1
SCHEMBL7409600 0.84 MAPT (0.42) PKMALDH1A1SMN1; SMN2RAB9A
SCHEMBL7466483 0.84 NPC1 (0.45) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL7380572 0.84 ITGB3 (0.40) SLC7A5NOS3NOS1NOS2ITGB3
SCHEMBL7382269 0.83 NR1H4 (0.41) ITGB3ITGAVITGA2BF2ALDH1A1
SCHEMBL7376793 0.83 RAB9A (0.38) ITGB3ITGA2BF2ALDH1A1SMN1; SMN2
SCHEMBL7410561 0.82 ITGB3 (0.40) SLC7A5ITGB3ITGAVITGA2BITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP claimed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed